| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DHODH |
2-aminoethanol;5-[4-(6-carboxynaphthalen-2-yl)butyl]-2,4-dioxo-1H-pyrimidine-6-carboxylic acid |
986000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
US10968216, Example 293 |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
N-(2,2-Diphenylethyl)-4-hydroxy-1,2,5-thiadiazole-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
3-(5-Cyclopropylpyrimidin-2-yl)-1-[(2-fluorophenyl)methyl]pyrazolo[3,4-b]pyridine |
NA |
313800 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
2-(4-Pyrimidin-5-ylphenyl)quinoline-4-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
Methyl 2-(4-cyclohexylphenyl)quinoline-4-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
2-(4-Morpholin-4-ylphenyl)quinoline-4-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
Methyl 2-(4-pyridin-3-ylphenyl)quinoline-4-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
2-(4-Pyrimidin-2-ylphenyl)quinoline-4-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
Methyl 2-(4-piperidin-1-ylphenyl)quinoline-4-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-benzyl-4-oxo-1,2,5-thiadiazole-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
2-methyl-3-[(N-methylanilino)methyl]-5-oxo-1H-pyrazole-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
2-methyl-5-oxo-3-(phenoxymethyl)-1H-pyrazole-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-4-oxo-1,2,5-oxadiazole-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
2-methyl-5-oxo-3-(phenylsulfanylmethyl)-1H-pyrazole-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
3-(anilinomethyl)-2-methyl-5-oxo-1H-pyrazole-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
2-(4-Chlorophenyl)-3-hydroxy-8-methoxyquinoline-4-carboxylicacid |
NA |
306000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHODH |
2-(4-Chlorophenyl)-3-hydroxy-7-methoxyquinoline-4-carboxylate |
NA |
151000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHODH |
2-(4-Chlorophenyl)-3-hydroxy-8-trifluoromethylquinoline-4-carboxylic acid |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHODH |
2-(4-Chlorophenyl)-3-hydroxy-8-methylquinoline-4-carboxylicacid |
NA |
212000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |