| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DHODH |
3-(5-Cyclopropylpyrimidin-2-yl)-1-[(2,6-dichlorophenyl)methyl]pyrrolo[2,3-b]pyridine |
NA |
340100 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
5-Cyclopropyl-2-[1-[(2,6-difluorophenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-4-amine |
NA |
177400 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
1-[(2-Chlorophenyl)methyl]-3-(5-cyclopropylpyrimidin-2-yl)pyrrolo[2,3-b]pyridine |
NA |
239800 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
1-[(2-Bromophenyl)methyl]-3-(5-cyclopropylpyrimidin-2-yl)pyrrolo[2,3-b]pyridine |
NA |
324400 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
3-(5-Cyclopropylpyrimidin-2-yl)-1-[(2-fluorophenyl)methyl]indazole |
NA |
546600 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
3-(5-Cyclopropylpyrimidin-2-yl)-1-(naphthalen-1-ylmethyl)pyrrolo[2,3-b]pyridine |
NA |
829100 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
3-(5-Cyclopropylpyrimidin-2-yl)-1-[(2,6-difluorophenyl)methyl]pyrrolo[2,3-b]pyridine |
NA |
172600 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
1-[(2-Bromo-6-chlorophenyl)methyl]-3-(5-cyclopropylpyrimidin-2-yl)pyrrolo[2,3-b]pyridine |
NA |
277900 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
3-(5-Cyclopropylpyrimidin-2-yl)-1-[(2,3-difluorophenyl)methyl]pyrrolo[2,3-b]pyridine |
NA |
248500 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
1-Benzyl-3-(5-cyclopropylpyrimidin-2-yl)pyrrolo[2,3-b]pyridine |
NA |
290900 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
3-(5-Cyclopropylpyrimidin-2-yl)-1-[(2,4,6-trifluorophenyl)methyl]pyrrolo[2,3-b]pyridine |
NA |
368200 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
3-Carbamoyl-5-[4-(4-methylphenyl)phenyl]benzoic acid |
100000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2-naphthyl)-5-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
5,6-dimethyl-N-(2-naphthyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-benzyl-5-methyl-N-(2-naphthyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
4-({5-Methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}amino)benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)quinolin-6-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
2-Methyl-7-[(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]chromen-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-anthracen-2-yl-5-methyl[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
5-ethyl-N-(2-naphthyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |