| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DHODH |
N,5-dimethyl-N-(2-naphthyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)quinolin-3-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(3-chloro-4-fluorophenyl)-2-methyl-3-nitrobenzamide |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
3-Carbamoyl-5-(3,5-diphenylphenyl)benzoic acid |
100000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
diethyl 2-[(1H-benzimidazol-5-ylamino)methylene]malonate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
Methyl 2-(4-phenylphenyl)quinoline-4-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
5-methyl-N-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
5-methyl-N-(naphthalen-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
1-(4-Chlorophenyl)-3-quinolin-8-ylurea |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
5-methyl-N-(1-naphthyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
1-(2-Methoxyphenyl)-3-naphthalen-1-ylurea |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
2-methyl-3-nitro-N-[3-(trifluoromethyl)phenyl]benzamide |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
3-[(5-Methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]naphthalen-2-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(3-bromophenyl)-2-methyl-3-nitrobenzamide |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
N-(3,5-dichlorophenyl)-2-methyl-3-nitrobenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
N-(4-bromo-2-methylphenyl)-2-naphthamide |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
Cinchophen |
NA |
144000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| DHODH |
N-(3,4-difluorophenyl)-2-methyl-3-nitrobenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
N-(2,2-diphenylethyl)-2-hydroxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
3-chloro-N-(2,2-diphenylethyl)-2-hydroxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |