| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DLG4 |
5-hydroxy-3-methyl-1H-indole-2,6-dicarboxylic acid |
530000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DLG4 |
(2S)-2-[[(2S)-2-[4-[(1R,2R)-1-amino-2-hydroxypropyl]triazol-1-yl]propanoyl]amino]-3-methylbutanoic acid |
289000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DLG4 |
(2S)-2-[4-[(1S)-1-[[(2S,3R)-2-amino-3-hydroxybutanoyl]amino]ethyl]triazol-1-yl]-3-methylbutanoic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DLG4 |
(S)-2-{(S)-2-[(S)-2-((S)-2-Amino-4-carbamoyl-butyrylamino)-3-hydroxy-propionylamino]-3-carboxy-propionylamino}-3-methyl-butyric acid |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DLG4 |
H-Glu-xiThr-Ala-Val-OH |
260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DLG4 |
(S)-4-amino-5-((S)-1-((S)-3-carboxy-1-((S)-1-carboxypropylamino)-1-oxopropan-2-ylamino)-3-hydroxy-1-oxopropan-2-ylamino)-5-oxopentanoic acid |
230000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DLG4 |
(S)-4-amino-5-((S)-1-((S)-3-carboxy-1-((S)-1-carboxy-2,2-dimethylpropylamino)-1-oxopropan-2-ylamino)-3-hydroxy-1-oxopropan-2-ylamino)-5-oxopentanoic acid |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DLG4 |
H-Gln-Thr-Ala-Val-OH |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DLG4 |
(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-(2-cyclohexylethylamino)-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-3-methylbutanoic acid |
141000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DLG4 |
naphth-2-ylethyl-Glu-Thr-Asp-Val-OH |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DLG4 |
(4S)-5-[[(2S,3R)-1-[[(2S)-3-carboxy-1-[[(1S)-1-carboxy-2-methylpropyl]amino]-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-4-[2-(3,4-dichlorophenyl)ethylamino]-5-oxopentanoic acid |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DLG4 |
naphth-2-ylethyl-Ala-Thr-Ala-Val-OH |
280000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DLG4 |
Me-Glu-thionoThr-Ala-Val-OH |
220000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DNASE1 |
4-[(4,6-Dichloro-1,3,5-triazin-2-yl)amino]-2-(3-hydroxy-6-oxoxanthen-9-yl)benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| DNM1 |
2,5-Bis(benzylamino)benzo-1,4-quinone |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| DNM1 |
4-[[4-(4-Carboxyanilino)-3,6-dioxocyclohexa-1,4-dien-1-yl]amino]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| DNM1 |
2-[[4-(2-Carboxyanilino)-3,6-dioxocyclohexa-1,4-dien-1-yl]amino]benzoic acid |
NA |
162000 |
NA |
NA |
NA |
NA |
BindingDB |
| DNM2 |
|
NA |
1300000 |
NA |
NA |
NA |
NA |
BindingDB |
| DNM2 |
4-Chloro-2-[[2-(4-hydroxyphenyl)-1,3-dioxoisoindole-5-carbonyl]amino]benzoic acid |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB |
| DNMT1 |
S-Inosyl-L-homocysteine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |