| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DHODH |
4-chloro-N-(2,2-diphenylethyl)-2-hydroxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
5-chloro-N-(2,2-diphenylethyl)-2-hydroxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
3,5-dichloro-N-(2,2-diphenylethyl)-2-hydroxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
5-bromo-N-(2,2-diphenylethyl)-2-hydroxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-3-fluoro-2-hydroxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-3,4-difluoro-2-hydroxybenzamide |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-2-hydroxy-5-methylbenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-2-hydroxy-3-methoxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-2-hydroxy-4-methoxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-2-hydroxy-5-methoxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-2-hydroxy-3-(hydroxymethyl)benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-2-hydroxy-4-(hydroxymethyl)benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-2-hydroxy-5-(hydroxymethyl)benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
N-(2,2-diphenylethyl)-4-formyl-2-hydroxybenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DHODH |
Bay 41-2272 |
NA |
351200 |
NA |
NA |
NA |
NA |
BindingDB |
| DHODH |
Vidofludimus |
NA |
232000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHRS9 |
(2S)-2-(hydroxymethyl)-2-methylchromen-6-ol |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB |
| DLG4 |
Ser-Ala-Val |
229000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DLG4 |
1-(3-Carboxypropyl)-3-methyl-5-phenylmethoxyindole-2,6-dicarboxylic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DLG4 |
(2S)-2-[[1-[(1S)-1-carboxy-2-methylpropyl]triazole-4-carbonyl]amino]-3-methylbutanoic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |