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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
EGFR N-(3-bromophenyl)-6-(2,5-dimethoxybenzyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 300000 NA NA NA NA TTD
EGFR N-(3-bromophenyl)-6-(2,4-dichlorobenzyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 300000 NA NA NA NA TTD
EGFR 6-(2,4-dichlorobenzyl)-N-(3-ethynylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 300000 NA NA NA NA TTD
EGFR N-(3-bromophenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 200000 NA NA NA NA TTD
EGFR N-(3-ethynylphenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 200000 NA NA NA NA TTD
EGFR 6-(2-Phenylethyl)-N-[3-(trifluoromethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 200000 NA NA NA NA TTD
EGFR N-(3-bromo-4-fluorophenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 200000 NA NA NA NA TTD
EGFR N-[4-fluoro-3-(trifluoromethyl)phenyl]-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 200000 NA NA NA NA TTD
EGFR N-(4-chloro-2-fluorophenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA 200000 NA NA NA NA TTD
EGFR 2-Amino-4-(m-bromoanilino)-6-benzyl-7-methyl-pyrrolo-[2,3-d]pyrimidine NA 200000 NA NA NA NA TTD
EGFR 4-N-(3-bromophenyl)-6-[(2,5-dimethoxyphenyl)methyl]-4-N-methyl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine NA 143500 NA NA NA NA BindingDB|TTD
EGFR Phloretin NA 25000000 NA NA NA NA BindingDB|PubChem|TTD
EGFR 4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol 296000 NA NA NA NA NA BindingDB|TTD
EGFR 2-[(4-Hydroxyphenyl)methylidene]propanedioic acid NA 1500000 NA NA NA NA BindingDB|TTD
EGFR Quercetin NA 190000 NA NA NA NA BindingDB|PubChem
EGFR Biochanin A NA 105000 NA NA NA NA BindingDB
EGFR Acacetin NA 140000 NA NA NA NA BindingDB
EGFR Apigenin NA 111000 NA NA NA NA BindingDB
EGFR 2-Amino-4-(N-methyl-m-bromoanilino)-6-benzyl-7-methyl-pyrrolo[2,3-d]pyrimidine NA 253600 NA NA NA NA BindingDB|TTD
EGFR N-(3-chlorobenzyl)benzofuro[2,3-b]pyridin-4-amine 1000000 NA NA NA NA NA TTD