Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| EGFR | (2E)-2-cyano-3-(4-nitrophenyl)prop-2-enoic acid | NA | 1300000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | benzylidenemalononitrile (BMN) deriv. 33 | 264000|NA | 700000|264000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | alpha-Cyano-4-hydroxycinnamic acid | NA|165000|308000 | 200000|308000|165000|NA | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| EGFR | 2-(1-(4-Aminophenyl)ethylidene)propanedinitrile | NA | 1250000 | NA | NA | NA | NA | TTD |
| EGFR | benzylidenemalononitrile (BMN) deriv. 38 | 341000 | 1100000|NA | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | (2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide | NA | 800000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | benzylidenemalononitrile (BMN) deriv. 40 | 360000 | 625000|NA | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | benzylidenemalononitrile (BMN) deriv. 41 | NA | 500000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | 2-[Hydroxy-(4-methoxyphenyl)methylidene]propanedinitrile | NA | 450000 | NA | NA | NA | NA | TTD |
| EGFR | 2-(Hydroxy(4-Hydroxyphenyl)Methylene)Malononitrile | NA | 230000 | NA | NA | NA | NA | TTD |
| EGFR | 2-cyano-3-(1H-pyrrol-2-yl)acrylic acid | NA | 1360000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | p-Hydroxycinnamonitrile | NA | 2400000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | Propanedinitrile, [(4-hydroxyphenyl)hydrazono]- | NA | 225000 | NA | NA | NA | NA | TTD |
| EGFR | 2-[(4-Hydroxyanilino)methylidene]propanedinitrile | NA | 350000 | NA | NA | NA | NA | TTD |
| EGFR | 2-(2,4,6-Trioxo-1,3-diazinan-5-ylidene)propanedinitrile | NA | 1400000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | Tyrphostin deriv. 71 | NA | 1000000 | NA | NA | NA | NA | TTD |
| EGFR | Sunitinib | NA | 172100 | NA | NA | NA | NA | BindingDB|PubChem |
| EGFR | Dimeric Tyrphostin 11 | NA | 112000 | NA | NA | NA | NA | BindingDB |
| EGFR | 2-Benzoyl-3-(1H-indol-3-yl)propenenitrile | NA | 300000 | NA | NA | NA | NA | BindingDB |
| EGFR | Methyl 2,5-dihydroxycinnamate | NA | 102000 | NA | NA | NA | NA | BindingDB |