Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| EGFR | 4-N-(3-bromophenyl)-7-[(2-methylphenyl)methyl]pyrrolo[2,3-d]pyrimidine-2,4-diamine | NA | 113300 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | 4-N-(3-bromophenyl)-7-[(3,4-dichlorophenyl)methyl]pyrrolo[2,3-d]pyrimidine-2,4-diamine | NA | 200000 | NA | NA | NA | NA | TTD |
| EGFR | Aztreonam | NA | NA | NA | NA | NA | 400000 | PubChem |
| EGFR | US9422297, Aag145-344 | NA | 232700 | NA | NA | NA | NA | BindingDB |
| EGFR | Levodopa | NA | 900000 | NA | NA | NA | NA | PubChem|TTD |
| EGFR | Adenosine | NA | 195000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| EGFR | p-Coumaric acid | 1000000 | 3000000|NA | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | 2-[(1-Oxidopyridin-1-ium-4-yl)methylidene]propanedinitrile | NA | 1300000 | NA | NA | NA | NA | TTD |
| EGFR | 2-((3,5-Dimethyl-4-hydroxyphenyl)-methylene)-4-cyclopentene-1,3-dione | NA | 440000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | alpha-Cyanocinnamic acid | 850000|NA | NA|850000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | Marein | NA | 19000000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | Pelitinib | NA | 83000000 | NA | NA | NA | NA | BindingDB |
| EGFR | Carumonam | NA | NA | NA | NA | NA | 500000 | PubChem |
| EGFR | 3'-Chloro-5,7-dimethoxyisoflavone | NA | 500000 | NA | NA | NA | NA | BindingDB |
| EGFR | Caffeic Acid | NA|400000 | 1000000|1200000|NA | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| EGFR | Propanedinitrile, [(3-hydroxy-4-methoxyphenyl)methylene]- | NA | 250000 | NA | NA | NA | NA | TTD |
| EGFR | N-[4-(3-bromoanilino)-3-cyanoquinolin-6-yl]-4-(propylamino)but-2-ynamide | NA | 130017|130016.96 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | 2-[(6-nitro-2H-1,3-benzodioxol-5-yl)methylidene]propanedinitrile | NA | 560000 | NA | NA | NA | NA | BindingDB|TTD |
| EGFR | 2-{[4-(Methylsulfanyl)phenyl]methylidene}propanedinitrile | NA | 625000 | NA | NA | NA | NA | TTD |
| EGFR | Osimertinib | NA | 480000 | NA | NA | NA | NA | BindingDB|PubChem |