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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
EGLN1 3-[[(4-Hydroxy-7-phenoxy-3-isoquinolinyl)carbonyl]amino]-3-methylbutanoic acid NA 191920 NA NA NA NA BindingDB
EGLN1 3-[[7-(4-Fluorophenyl)-4-hydroxyisoquinoline-3-carbonyl]amino]-2,2-dimethylpropanoic acid NA 113830 NA NA NA NA BindingDB
EGLN1 4-[[(4-methylphenyl)sulfonyl]oxy]Cyclohexanecarboxylic acid NA 200000 NA NA NA NA BindingDB
EGLN1 3-{[4-Hydroxy-7-(4-methoxy-benzylamino)-isoquinoline-3-carbonyl]amino}-2,2-dimethyl-propionic acid NA 200000 NA NA NA NA BindingDB
EGLN1 3-[(1-Cyano-4-hydroxy-2-oxido-7-phenoxyisoquinolin-2-ium-3-carbonyl)amino]-2,2-dimethylpropanoic acid NA 200000 NA NA NA NA BindingDB
EGLN1 4-[(4-Hydroxy-7-phenoxy-isoquinoline-3-carbonyl)-amino]-2,2-dimethyl-butyric acid NA 118550 NA NA NA NA BindingDB
EGLN1 5-{[4-Hydroxy-7-(4-methoxy-benzylamino)-isoquinoline-3-carbonyl]amino}-pentanoic acid NA 158180 NA NA NA NA BindingDB
EGLN1 5-[[7-(2,6-Difluorophenoxy)-4-hydroxyisoquinoline-3-carbonyl]amino]pentanoic acid NA 200000 NA NA NA NA BindingDB
EGLN1 NA 111450 NA NA NA NA BindingDB
EGLN1 4-[[7-[(4-Fluorobenzoyl)amino]-4-hydroxyisoquinoline-3-carbonyl]amino]butanoic acid NA 200000 NA NA NA NA BindingDB
EGLN1 1-benzyl-8-hydroxy-2-oxo-N-(tetrazolidin-5-ylmethyl)-1,6-naphthyridine-7-carboxamide NA 138000 NA NA NA NA BindingDB
EGLN1 NA 200000 NA NA NA NA BindingDB
EGLN1 2-[(3-Hydroxypyridin-2-yl)formamido]acetic acid NA 409000 NA NA NA NA BindingDB
EGLN2 (1-Hydroxy-2,5-dioxo-pyrrolidin-3-yl)-acetic acid NA 1000000 NA NA NA NA BindingDB|TTD
EGLN2 Salicyluric Acid NA 1000000 NA NA NA NA PubChem|TTD
EGLN2 2,4-Pyridinedicarboxylic acid NA 624800 NA NA NA NA BindingDB
EGLN2 Succinic Acid NA 830000 NA NA NA NA BindingDB|PubChem
EGLN2 2-((Pyridin-2-yl)formamido)acetic acid NA 1000000 NA NA NA NA TTD
EGLN2 2-(3-Hydroxyphenyl)-2-oxo-ethanoic acid NA 1000000 NA NA NA NA TTD
EGLN2 Citric Acid NA 6300000 NA NA NA NA BindingDB|PubChem