| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| EGLN2 |
Fumaric Acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| EGLN2 |
Malic Acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
PubChem |
| EGLN2 |
2-(3-Hydroxyphenyl)-2-mercaptoacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGLN2 |
Isocinchomeronic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EGLN3 |
Succinic Acid |
NA |
570000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| EGLN3 |
Citric Acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| EGLN3 |
Malic Acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
PubChem |
| EHMT1 |
(2R,3S,4R,5R)-2-[(2R)-2-amino-3-cyclopropylpropyl]-5-(6-aminopurin-9-yl)oxolane-3,4-diol |
NA |
794300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT1 |
(2R,3S,4R,5R)-2-[(2S)-2-amino-3-cyclohexylpropyl]-5-(6-aminopurin-9-yl)oxolane-3,4-diol |
NA |
203700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT1 |
(2R,3S,4R,5R)-2-[(2R)-2-amino-3-cyclobutylpropyl]-5-(6-aminopurin-9-yl)oxolane-3,4-diol |
NA |
115000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT1 |
(2R,3S,4R,5R)-2-[(2R)-2-amino-3-cyclohexylpropyl]-5-(6-aminopurin-9-yl)oxolane-3,4-diol |
NA |
145800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT1 |
(2S,5R)-2,5-diamino-6-[(2S,3R,4S,5S)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]hexanoic acid |
NA |
513000 |
NA |
NA |
NA |
NA |
BindingDB |
| EHMT1 |
N-[3-[(2-amino-6-methylpyrimidin-4-yl)amino]phenyl]-4-(quinolin-4-ylamino)benzamide |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT1 |
Sinefungin |
NA |
513000 |
NA |
NA |
NA |
NA |
BindingDB |
| EHMT1 |
N-[2-[(2-amino-6-methylpyrimidin-4-yl)amino]phenyl]-3-(quinolin-4-ylamino)benzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT1 |
N-[2-[(2-amino-6-methylpyrimidin-4-yl)amino]phenyl]-4-(quinolin-4-ylamino)benzamide |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT1 |
(2R,3R,4S,5R)-2-(6-aminopurin-9-yl)-5-(3-phenylpropyl)oxolane-3,4-diol |
NA |
235000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT1 |
(2R,3S,4R,5R)-2-[2-amino-3-(3,4-dimethoxyphenyl)propyl]-5-(6-aminopurin-9-yl)oxolane-3,4-diol |
NA |
147000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EHMT2 |
(2R,3S,4R,5R)-2-[(2S)-2-amino-3-cyclobutylpropyl]-5-(6-aminopurin-9-yl)oxolane-3,4-diol |
NA |
169000 |
NA |
NA |
NA |
NA |
TTD |
| EHMT2 |
(2R,3S,4R,5R)-2-[(2S)-2-amino-3-cyclopentylpropyl]-5-(6-aminopurin-9-yl)oxolane-3,4-diol |
NA |
191300 |
NA |
NA |
NA |
NA |
TTD |