| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| EHMT2 |
(2R,3S,4R,5R)-2-[2-amino-3-(3,4-dimethoxyphenyl)propyl]-5-(6-aminopurin-9-yl)oxolane-3,4-diol |
NA |
157000 |
NA |
NA |
NA |
NA |
TTD |
| EIF2AK2 |
N-[5-(6,7-dimethoxyquinolin-4-yl)oxypyridin-2-yl]-1-methyl-3-oxo-2,5-diphenylpyrazole-4-carboxamide |
NA |
480000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EIF2AK4 |
1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- |
470000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF2AK4 |
Motesanib |
4400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF2AK4 |
Erlotinib |
4400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF2AK4 |
Dasatinib |
1600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF2AK4 |
Sunitinib |
180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF2AK4 |
Jnj-7706621 |
3900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF2AK4 |
Tozasertib |
1900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF2AK4 |
Pelitinib |
290000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF2AK4 |
|
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
2-[5-(4-Butylphenyl)furan-2-yl]-6-methylquinoline-4-carboxylic acid |
NA |
105100 |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
6-Bromo-2-[5-(4-butylphenyl)furan-2-yl]quinoline-4-carboxylic acid |
NA |
160600 |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
2-[5-(4-Butylphenyl)furan-2-yl]-6-phenylquinoline-4-carboxylic acid |
NA |
124300 |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
2-[5-(4-Butylphenyl)furan-2-yl]-6-propan-2-ylquinoline-4-carboxylic acid |
NA |
107300 |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
2-[5-(4-Butylphenyl)furan-2-yl]-6,8-dimethylquinoline-4-carboxylic acid |
NA |
111300 |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
2-[5-(4-Butylphenyl)furan-2-yl]-6-ethylquinoline-4-carboxylic acid |
NA |
146600 |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
Ethyl 6-bromo-2-[5-(4-butylphenyl)furan-2-yl]quinoline-4-carboxylate |
NA |
129100 |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
2-[5-(4-Butylphenyl)furan-2-yl]-5-chloroquinoline-4-carboxylic acid |
NA |
135400 |
NA |
NA |
NA |
NA |
BindingDB |
| EIF4A1 |
6-Acetamido-2-[5-(4-butylphenyl)furan-2-yl]quinoline-4-carboxylic acid |
NA |
125800 |
NA |
NA |
NA |
NA |
BindingDB |