| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ELANE |
(S)-2-[(S)-2-(3,3-Dimethyl-butanoylamino)-3,3-dimethyl-butanoylamino]-N4,N4-dimethyl-N1-[1-methyl-2-(5-methyl-benzoxazol-2-yl)-2-oxo-ethyl]-succinamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
(S)-N1-((S)-3-Benzylcarbamoyl-3,3-difluoro-1-methyl-2-oxo-propyl)-2-[(S)-2-(3,3-dimethyl-butanoylamino)-3,3-dimethyl-butanoylamino]-N4,N4-dimethyl-succinamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
(2S)-2-[[(2S)-2-(3,3-dimethylbutanoylamino)-3,3-dimethyl-butanoyl]amino]-N',N'-dimethyl-N-(1-methyl-2-oxazolo[4,5-b]pyridin-2-yl-2-oxo-ethyl)butanediamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
[4-[[2-[(E)-C-ethyl-N-hydroxycarbonimidoyl]phenyl]sulfamoyl]phenyl] 2,2-dimethylpropanoate |
NA |
679370 |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
[4-[[2-[(E)-N-hydroxy-C-propylcarbonimidoyl]phenyl]sulfamoyl]phenyl] 2,2-dimethylpropanoate |
NA |
367500 |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
[4-[[2-[(E)-hydroxyiminomethyl]phenyl]sulfamoyl]phenyl] 2,2-dimethylpropanoate |
NA |
394440 |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
[4-[[2-[(E)-N-methoxy-C-methylcarbonimidoyl]phenyl]sulfamoyl]phenyl] 2,2-dimethylpropanoate |
NA |
323890 |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
[4-[[2-[(Z)-N-methoxy-C-methylcarbonimidoyl]phenyl]sulfamoyl]phenyl] 2,2-dimethylpropanoate |
NA |
367180 |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
[4-[[2-[(E)-N-(3-hydroxypropoxy)-C-methylcarbonimidoyl]phenyl]sulfamoyl]phenyl] 2,2-dimethylpropanoate |
NA |
158800 |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
trans-Epoxysuccinyl-L-leucylamido-(4-guanidino)butane |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
3-Acetoxymethyl-7,7-dibromo-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester |
NA |
1390000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
Tetrasodium;[4-[4-oxo-5-[[3-[[4-oxo-7-sulfonatooxy-2-(4-sulfonatooxyphenyl)chromen-5-yl]oxymethyl]phenyl]methoxy]-7-sulfonatooxychromen-2-yl]phenyl] sulfate |
NA |
157000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
Xeruborbactam |
NA |
132000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| ELANE |
4-((2S,3S)-3-Ethyl-4-oxo-azetidin-2-yloxy)-benzoic acid |
290000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
(S)-2-((S)-2-(3,3-dimethylbutanamido)-3,3-dimethylbutanamido)-N4,N4-dimethyl-N1-(4,4,4-trifluoro-3-oxobutan-2-yl)succinamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
tert-butyl N-[(2S)-1-[(2S)-2-[(1-diphenoxyphosphoryl-2,2-dimethylpropyl)carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
Boc-Val-Pro-DL-Nva-thiazol-2-yl |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
3-Acetoxymethyl-7,8-dioxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
6,7-dimethoxy-2-methyl-4H-3,1-benzoxazin-4-one |
794300|831763.77 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
benzhydryl (7Z)-3-(acetyloxymethyl)-8-oxo-7-(pyridin-2-ylmethylidene)-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |