| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ELANE |
[3,5-Dibutyl-2-oxo-6-(2-oxopropyl)pyran-4-yl] acetate |
288403|288403.15 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
[3,5-Dibutyl-2-(3-methyloxiran-2-yl)-6-oxopyran-4-yl] acetate |
338844|338844.16 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
[3,5-Dibutyl-2-(2-hydroxypropyl)-6-oxopyran-4-yl] acetate |
346737|346736.85 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
Met-Phe-Leu-Glu-Ala-Ile-Pro-Met |
270000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
3-({1-[2-(2-tert-Butoxycarbonylamino-propionylamino)-propionyl]-pyrrolidine-2-carbonyl}-amino)-2,2-difluoro-4-methyl-pentanoic acid ethyl ester |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
2-[(Imidazole-1-carbonyl)-amino]-pentanoic acid methyl ester |
320000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
2-[(Imidazole-1-carbonyl)-amino]-3-methyl-butyric acid methyl ester |
1800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
2-[(Imidazole-1-carbonyl)-amino]-hexanoic acid methyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
(R)-3-Methyl-7-oxo-4-thia-1-aza-bicyclo[3.2.0]hept-2-ene-2-carboxylic acid benzyl ester |
310000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
3-Acetoxymethyl-8-oxo-7-vinylidene-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester |
NA |
9000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
CID 44342779 |
NA |
13500000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
CID 44342794 |
NA |
5400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
(R)-3-Acetoxymethyl-7-amino-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydryl ester |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
benzhydryl (7Z)-3-(acetyloxymethyl)-5,5,8-trioxo-7-(2-oxopropylidene)-5lambda6-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
benzhydryl (7Z)-3-(acetyloxymethyl)-7-(2-methoxy-2-oxoethylidene)-5,5,8-trioxo-5lambda6-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate |
NA |
8900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
benzhydryl (7Z)-3-(acetyloxymethyl)-7-[2-[methoxy(methyl)amino]-2-oxoethylidene]-5,5,8-trioxo-5lambda6-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
benzhydryl (7Z)-3-(acetyloxymethyl)-7-(2-methoxy-2-oxoethylidene)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate |
NA |
2600000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
benzhydryl (7Z)-3-(acetyloxymethyl)-7-(2-hydroxyethylidene)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
benzhydryl (7Z)-3-(acetyloxymethyl)-7-benzylidene-5,5,8-trioxo-5lambda6-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate |
NA |
8900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |