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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ERAP1 2-[[[1-Amino-2-(2-methylpropylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acid 250000 NA NA NA NA NA TTD
ERAP1 2-[[[1-Amino-2-(cyclohexylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-(oxolan-2-ylmethylamino)ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 (1-Amino-2-piperidin-1-ylethyl)phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-[(2-aminocyclohexyl)amino]ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-(1-phenylethylamino)ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-[2-(dimethylamino)ethylamino]ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 2-Benzyl-3-[1,2-diaminoethyl(hydroxy)phosphoryl]propanoic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-(cycloheptylamino)ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-(2-phenylethylamino)ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 2-[[[1-Amino-2-(propylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-(2-piperazin-1-ylethylamino)ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-[(4-tert-butylphenyl)methylamino]ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-[(4-aminophenyl)methylamino]ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 2-[[[1-Amino-2-(cycloheptylamino)ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-[(4-methoxyphenyl)methylamino]ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 2-[[[1-Amino-2-[2-(4-methoxyphenyl)ethylamino]ethyl]-hydroxyphosphoryl]methyl]-3-phenylpropanoic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-(hexylamino)ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-[[4-(aminomethyl)phenyl]methylamino]ethyl]phosphonic acid 250000 NA NA NA NA NA TTD
ERAP1 [1-Amino-2-[2-(4-methoxyphenyl)ethylamino]ethyl]phosphonic acid 250000 NA NA NA NA NA GtoPDB|TTD