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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
EPHX2 2-(1-methyl-1H-pyrazol-4-yl)-1H-benzimidazole NA 127000 NA NA NA NA ChEMBL|TTD
EPHX2 Fuberidazole NA 207000 NA NA NA NA TTD
EPHX2 N-Cyclohexyl-N'-(3-hydroxypropyl)urea NA 500000 NA NA NA NA TTD
EPHX2 Celecoxib NA 261140 NA NA NA NA PubChem
EPHX2 3-(4-(Benzyloxy)phenyl)propan-1-ol NA 150000 NA NA NA NA ChEMBL|TTD
EPHX2 1-[3-(Trifluoromethyl)pyridin-2-yl]piperazine NA 1200000 NA NA NA NA ChEMBL|TTD
EPHX2 N-[2-(morpholin-4-yl)phenyl]thiophene-3-carboxamide NA 171000 NA NA NA NA ChEMBL|TTD
EPHX2 Sodium Lauryl Sulfate NA 300000|101000 NA NA NA NA PubChem
EPHX2 N-((Cyclohexylamino)carbonyl)glycine NA 500000 NA NA NA NA TTD
EPHX2 1-Cyclohexyl-3-(5-hydroxy-pentyl)-urea NA 253000 NA NA NA NA TTD
EPHX2 Boc-3-amino-1,2,3,4-tetrahydroquinoline NA 580000 NA NA NA NA ChEMBL|TTD
EPHX2 4-(2,5-dimethyl-1-((oxolan-2-yl)methyl)-1H-pyrrol-3-yl)-1,3-thiazol-2-amine NA 195000 NA NA NA NA ChEMBL|TTD
EPHX2 Oxaprozin NA 300000 NA NA NA NA PubChem
EPHX2 1-Methyl-N-(2-phenylethyl)-1H-pyrazole-3-methanamine NA 8e+05|800000 NA NA NA NA ChEMBL|TTD
EPHX2 N-Methyl-N-(3-pyridin-3-ylbenzyl)amine NA 2200000 NA NA NA NA ChEMBL|TTD
EPHX2 2-(Furan-2-yl)benzo[d]oxazole NA 133000 NA NA NA NA TTD
EPOR (S)-2-{Bis-[(E)-3-(3-phenoxy-phenyl)-allyl]-amino}-3-hydroxy-propionic acid methyl ester NA 145000 NA NA NA NA BindingDB|TTD
ERAP1 2-[[(1-Amino-3-phenylpropyl)-hydroxyphosphoryl]methyl]-3-(3,5-dimethylphenyl)propanoic acid 250000 NA NA NA NA NA TTD
ERAP1 methyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate NA 110000 NA NA NA NA BindingDB|TTD
ERAP1 (1-Amino-2-morpholin-4-ylethyl)phosphonic acid 250000 NA NA NA NA NA TTD