| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ESR2 |
N,N''-Diisobutyl-2-(2-naphthalen-1-yl-ethyl)-pyrimidine-4,6-diamine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ESR2 |
2-(3-methylbutyl)-4-N-(2-methylpropyl)-6-N-(naphthalen-1-ylmethyl)pyrimidine-4,6-diamine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ESR2 |
2,4-Diisobutylamino-pyrimidine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ESR2 |
N2,N4-bis(naphthalen-1-ylmethyl)-6-phenethylpyrimidine-2,4-diamine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ESR2 |
2,4-Diisobutylamino-6-chloropyrimidine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ESR2 |
3-(((6-((5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid |
NA |
NA |
NA |
534000 |
NA |
NA |
TTD |
| ESR2 |
Resorcinol |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| ESR2 |
2,2,2-Trifluoro-1-(6-methoxy-3,4-dihydroisoquinolin-2(1H)-yl)ethanone |
NA |
NA |
NA |
227000 |
NA |
NA |
ChEMBL|TTD |
| ESR2 |
Progesterone |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| ESR2 |
Miristalkonium chloride |
NA |
NA |
NA |
NA |
2818380|22387200 |
NA |
PubChem |
| ESR2 |
Phenol |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| ESRRA |
Scopolamine hydrobromide trihydrate |
NA |
NA |
NA |
NA |
217120 |
NA |
PubChem |
| ESRRA |
Miristalkonium chloride |
NA |
NA |
NA |
NA |
14125400|11220200|15848900 |
NA |
PubChem |
| EYA2 |
[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-[(4-methylpiperazin-1-yl)iminomethyl]-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate |
NA |
NA |
NA |
NA |
223872 |
NA |
PubChem |
| EYA2 |
Estradiol Valerate |
NA |
NA |
NA |
NA |
281838 |
NA |
PubChem |
| EYA2 |
Mebeverine Hydrochloride |
NA |
NA |
NA |
NA |
2511890 |
NA |
PubChem |
| EYA2 |
Acetarsol |
NA |
NA |
NA |
NA |
5623410 |
NA |
PubChem |
| EYA2 |
Dipyridamole |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| EYA2 |
Idarubicin |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| EYA2 |
Diclofenac sodium |
NA |
NA |
NA |
NA |
158489 |
NA |
PubChem |