| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| EYA2 |
Sodium Fluoride |
NA |
6600000 |
NA |
NA |
NA |
NA |
PubChem |
| EYA2 |
20-Hydroxyecdysone |
NA |
NA |
NA |
NA |
733271 |
NA |
PubChem |
| EYA2 |
Edetic Acid |
NA |
380000|1000000 |
NA |
NA |
NA |
NA |
PubChem |
| EZH2 |
N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-2-fluoro-3-methoxybenzamide |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| EZH2 |
(2S)-2-amino-4-[[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methylsulfanyl]-N-benzylbutanamide |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| EZH2 |
N-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-2-methylbenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| EZH2 |
N-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-2,3-dimethoxybenzamide |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
| EZH2 |
N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-methoxybenzamide |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-(2-Amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-2-[3-(4-fluoro-phenylmethanesulfonylamino)-6-methyl-2-oxo-2H-pyridin-1-yl]-acetamide |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
2-Chloro-benzenesulfonic acid 3-methyl-5-[2-(methyl-pyridin-4-yl-amino)-ethoxy]-phenyl ester |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-Acetylamino-N-[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-3-hydroxy-propionamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N'-hydroxy-3-[[[(6-methoxynaphthalen-2-yl)sulfonylamino]-(2-methylpiperidine-1-carbonyl)amino]methyl]benzenecarboximidamide |
111000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
3-[[azepane-1-carbonyl-[(6-methoxynaphthalen-2-yl)sulfonylamino]amino]methyl]-N'-hydroxybenzenecarboximidamide |
103000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(1-{[(4-Carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-2-hydroxy-ethyl)-carbamic acid tert-butyl ester |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(S)-1-(3,3-Diphenyl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA |
980000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(2S)-N-[(2S)-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-(1,2,3,4-tetrahydroquinoline-2-carbonyl)pyrrolidine-2-carboxamide |
NA |
660000 |
NA |
NA |
NA |
NA |
BindingDB |
| F10 |
5-Chloro-thiophene-2-carboxylic acid {(S)-3-methyl-1-[4-(3-oxo-morpholin-4-yl)-phenylcarbamoyl]-butyl}-amide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-(2,6-Difluoro-phenyl)-7-nitro-benzo[d][1,3]oxazin-4-one |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
5-Chloro-thiophene-2-carboxylic acid {[4-(3-oxo-morpholin-4-yl)-phenylcarbamoyl]-methyl}-amide |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(2S)-N-[(6-amino-2,4-dimethylpyridin-3-yl)methyl]-1-[(2R)-2-amino-3,3-diphenylpropanoyl]pyrrolidine-2-carboxamide |
240000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |