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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
F2 4-Chloro-N-(4-guanidino-phenyl)-2-hydroxy-benzamide 450000 NA NA NA NA NA TTD
F2 N-(4-Guanidino-phenyl)-2-hydroxy-5-methoxy-benzamide 450000 NA NA NA NA NA TTD
F2 3-Hydroxy-4-iodo-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide 310000 NA NA NA NA NA TTD
F2 4-Bromo-3-hydroxy-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide 330000 NA NA NA NA NA TTD
F2 3-Hydroxy-4-methoxy-anthracene-2-carboxylic acid (4-guanidino-phenyl)-amide 205000 NA NA NA NA NA TTD
F2 3-Hydroxy-4-iodo-anthracene-2-carboxylic acid (4-guanidino-phenyl)-amide 450000 NA NA NA NA NA TTD
F2 4-Bromo-3-hydroxy-anthracene-2-carboxylic acid (4-guanidino-phenyl)-amide 450000 NA NA NA NA NA TTD
F2 N-(4-Guanidino-phenyl)-2-hydroxy-3-iodo-5-methyl-benzamide 450000 NA NA NA NA NA TTD
F2 3-Hydroxy-anthracene-2-carboxylic acid (4-guanidino-phenyl)-amide 450000 NA NA NA NA NA TTD
F2 2-Hydroxy-biphenyl-3-carboxylic acid (4-guanidino-phenyl)-amide 450000 NA NA NA NA NA TTD
F2 3-Bromo-N-(4-guanidino-phenyl)-2-hydroxy-5-methyl-benzamide 125000 NA NA NA NA NA TTD
F2 3-Chloro-N-(4-guanidino-phenyl)-2-hydroxy-benzamide 450000 NA NA NA NA NA TTD
F2 N-(4-Guanidino-phenyl)-2-hydroxy-3-methyl-benzamide 450000 NA NA NA NA NA TTD
F2 (2S)-2-[[(2S)-2-amino-3-phenylpropanoyl]amino]-N-[(1R,2S)-3-cyclohexyl-1-hydroxy-1-(1,3-thiazol-2-yl)propan-2-yl]-4-methylpentanamide NA 530000 NA NA NA NA TTD
F2 [5-[4-[[4-(Aminomethyl)-1-bicyclo[2.2.2]octanyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(aminomethyl)-1-bicyclo[2.2.2]octanyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[(4-aminocyclohexyl)methylcarbamoyl]piperazine-1-carboxylate 274000 NA NA NA NA NA TTD
F2 [3-[[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxymethyl]-1-adamantyl]methyl 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 363000 NA NA NA NA NA TTD
F2 [5-[4-(6-Imidazol-1-ylhexanoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(6-imidazol-1-ylhexanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 [5-[4-(4-Piperidin-4-ylbutanoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(4-piperidin-4-ylbutanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
F2 N-[[4-(aminomethyl)phenyl]methyl]-N'-[[4-[[[4-[[4-(aminomethyl)phenyl]methylamino]-4-oxobutanoyl]amino]methyl]phenyl]methyl]butanediamide 1000000 NA NA NA NA NA TTD