GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ABCC2 |
Ketorolac Tromethamine |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Clarithromycin |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Nicotine |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Melatonin |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-24-[(2S)-1-[4-(2-methoxyethyl)piperazin-1-yl]propan-2-yl]-1,4,7,10,12,15,19,25,27,28-decamethyl-6,9,18-tris(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undecone |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
ABCC2 |
Lopinavir |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Aminophylline |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Oxiconazole Nitrate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Fluvoxamine Maleate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Thioacetazone |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Dexlansoprazole |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Gemifloxacin Mesylate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Galantamine |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Eszopiclone |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Procarbazine Hydrochloride |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Betamethasone |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Desmopressin Acetate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
17-Hydroxy-19-norpregn-4-en-20-yn-3-one |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
(R)-2-(3-(Diisopropylamino)-1-phenylpropyl)-4-methylphenol 2,3-dihydroxysuccinate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Fesoterodine Fumarate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |