Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| KCNE1 | Telbivudine | NA | 251189 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Etravirine | NA | 1258925|1258930 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Lapatinib | NA | 251189 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Alfuzosin | NA | 125893 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Darunavir | NA | 316228 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Lacosamide | NA | 251189 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Dasatinib | NA | 251189 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Lamotrigine | NA | 158489 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Sitagliptin | NA | 316228 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | 2-[2-ethoxy-5-(4-ethylpiperazin-1-yl)sulfonylphenyl]-5-methyl-7-propyl-2,3-dihydro-1H-imidazo[5,1-f][1,2,4]triazin-4-one | NA | 630957 | NA | NA | NA | NA | BindingDB |
| KCNE1 | NA | 158489|398107 | NA | NA | NA | NA | BindingDB | |
| KCNE1 | Silodosin | NA | 251189 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Nilotinib | NA | 398107 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Ambrisentan | NA | 501187 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Dofetilide | NA | 158489|251189 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNE1 | Doripenem | NA | 316228 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNH2 | (2-(2,4-Dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone | NA | 160000 | NA | NA | NA | NA | BindingDB |
| KCNH2 | Ecgonine methyl ester | NA | 416869.38 | NA | NA | NA | NA | BindingDB|TTD |
| KCNH2 | Tadalafil | NA | 125893 | NA | NA | NA | NA | BindingDB|PubChem |
| KCNH2 | 7-((R)-3-((S)-2-cyano-1-(methylamino)ethyl)pyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-8-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid | 150000 | NA | NA | NA | NA | NA | TTD |