| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
US10155727, Example 57 |
NA |
126000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
US10155727, Example 75 |
NA |
131000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
US10155727, Example 93 |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
US10155727, Example 94 |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
4-[3-(difluoromethoxy)-4-fluorophenyl]-1-(1H-pyrazol-5-ylmethyl)pyrazole |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
US10155727, Example 76 |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
US10155727, Example 101 |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
7-[3-(1-Aminocyclopropyl)pyrrolidin-1-yl]-1-cyclopropyl-6-fluoro-8-methyl-2-oxoquinoline-3-carboxylic acid |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
7-[(3R)-3-[(1S)-1-aminoethyl]pyrrolidin-1-yl]-1-cyclopropyl-6-fluoro-8-methyl-2-oxoquinoline-3-carboxylic acid |
NA |
214000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
US10081635, Example 5 |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
(1r)-1-[(4-{[(6,7-Dihydro[1,4]dioxino[2,3-C]pyridazin-3-Yl)methyl]amino}piperidin-1-Yl)methyl]-9-Fluoro-1,2-Dihydro-4h-Pyrrolo[3,2,1-Ij]quinolin-4-One |
NA |
238000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Methyl ecgonidine |
NA |
169824.37 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
2-[(2S)-2,3-dihydroxypropyl]-6-methoxy-1-oxo-4-phenyl-1,2-dihydroisoquinoline-3-carbonitrile |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
6-[[[1-[2-(2-oxo-7-pyrimidin-5-yloxy-1,8-naphthyridin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one |
NA |
224000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
Desvenlafaxine |
NA |
251189|19952623|19952600|251188.64 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
7-(1-Amino-3-azabicyclo[3.1.0]hexan-3-yl)-4-(aminomethyl)-1-cyclopropyl-6-fluoro-8-methylquinolin-2-one |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
US10508107, Example 17 |
NA |
518200 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
US10508107, Example 18 |
NA |
711500 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Azd-7648 |
NA |
198000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| KCNH2 |
US10407446, Example 9 |
NA |
198000 |
NA |
NA |
NA |
NA |
TTD |