| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
3-chloro-2-[(E)-2-(2-chlorophenyl)sulfonylethenyl]pyridine |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3-[(1S)-1-(2-amino-6,8-difluoroquinolin-3-yl)oxyethyl]-4-pyrazol-1-ylbenzoic acid |
NA |
144000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Levofloxacin |
NA |
912010.84|912011|915000|1100000|2100000|2300000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Moxifloxacin |
NA |
117489.76|117490|128824.96|128825|129000|398107 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| KCNH2 |
4-[3-[4-[(E)-2-(3-fluoropyridin-2-yl)ethenyl]sulfonylphenoxy]propyl]morpholine;hydrochloride |
NA |
112000|112100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
US10508107, Example 1 |
NA |
216600 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
N-[3-[(5-fluoro-2-oxo-1H-pyrimidin-6-yl)amino]-3-oxopropyl]-3-nitrobenzamide |
NA |
356180 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
3-nitro-N-[3-oxo-3-[(2-oxooxolan-3-yl)amino]propyl]benzamide |
NA |
904350 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
PqsR/LasR-IN-3 |
NA |
109010 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
7-(1-Amino-3-azabicyclo[3.1.0]hexan-3-yl)-4-(aminomethyl)-1-cyclopropyl-3,6-difluoro-8-methylquinolin-2-one |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Telbivudine |
NA |
5011872|158489319|5011870|158489000|5011872.34 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
N-(1-(1-isopropylpiperazine-4-carbonyl)piperidin-4-yl)cyclopentanecarboxamide |
NA |
156666.6667|156666.67 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
[4-(3-Aza-bicyclo[3.2.2]nonane-3-carbonyl)-piperidin-1-yl]-(4-isopropyl-piperazin-1-yl)-methanone |
NA |
115000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
N-(3,4-dichlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide |
NA |
2030000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
N-(3-chlorophenyl)-7-pyridin-4-yl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide |
NA |
8340000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
HIV-1 inhibitor-41 |
NA |
2687100 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
(12S)-8-[(3R)-3-(1-aminocyclopropyl)pyrrolidin-1-yl]-7-fluoro-12-methyl-2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxylic acid |
NA |
297000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
7-[(3R)-3-(1-aminocyclopropyl)pyrrolidin-1-yl]-1-cyclopropyl-6-fluoro-8-methyl-2-oxoquinoline-3-carboxylic acid |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
2-[7-[3-(1-aminocyclopropyl)pyrrolidin-1-yl]-1-cyclopropyl-6-fluoro-8-methyl-2-oxoquinolin-4-yl]-N,N-dimethylacetamide |
NA |
293000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
5-[[7-[3-(1-aminocyclopropyl)pyrrolidin-1-yl]-1-cyclopropyl-6-fluoro-8-methyl-2-oxoquinolin-4-yl]methyl]-3H-1,3,4-oxadiazol-2-one |
NA |
188000 |
NA |
NA |
NA |
NA |
BindingDB |