| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
(2S)-6-[(3aR,4R,7aS)-4-amino-1,3,3a,4,5,6,7,7a-octahydroisoindol-2-yl]-7-fluoro-2-methyl-12-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,10-tetraene-11-carboxylic acid |
NA |
127000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
N-hydroxy-4-[[4-(1-phenylethyl)piperazin-1-yl]methyl]benzamide |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
6-[[[1-[2-(2-oxo-7-pyridin-2-yloxy-1,8-naphthyridin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one |
NA |
155000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
(1R)-1-[2-(3,5-dichlorophenyl)pyridin-3-yl]-2,2-dipyridin-3-ylethanol |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
3-[[5-(3,4-dihydro-2H-pyrano[2,3-c]pyridin-6-ylmethylamino)-1,3-dioxan-2-yl]methyl]-5-fluoro-1,7-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7,9-tetraen-11-one |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3-[[5-(6,7-Dihydro-[1,4]oxathiino[2,3-c]pyridazin-3-ylmethylamino)-1,3-dioxan-2-yl]methyl]-5-fluoro-1-azatricyclo[6.3.1.04,12]dodeca-4,6,8(12),9-tetraen-11-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
N-[(3S,10R,13S)-17-(4-methoxyimidazol-1-yl)-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15-decahydro-1H-cyclopenta[a]phenanthren-3-yl]pyridazine-4-carboxamide |
NA |
856000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
5-amino-N-(2,6-dimethoxypyrimidin-4-yl)-1-[[4-(morpholin-4-ylmethyl)phenyl]methyl]triazole-4-carboxamide |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Dalfampridine |
NA |
4365158.32|4400000|4365160 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Phenytoin |
NA |
239883.29|240000|239883 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| KCNH2 |
Etravirine |
NA |
158489|398107 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| KCNH2 |
Lapatinib |
NA |
630957|100000000|630957.34 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Alfuzosin |
NA |
125893|125892.54 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Darunavir |
NA |
158489 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| KCNH2 |
Deferasirox |
NA |
3981070|3981071.71 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| KCNH2 |
Lacosamide |
NA |
50118723|50118700|50118723.36 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
2,6-Dioctylpyridine |
NA |
NA |
190546 |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3-Benzoyloxy-8-methyl-8-azabicyclo[3.2.1]octane-4-carboxylic acid |
NA |
3981071.71 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
(S)-4-((4-(((2,3-Dihydro-[1,4]dioxino[2,3-C]pyridin-7-Yl)methyl)amino)piperidin-1-Yl)methyl)-3-Fluoro-4-Hydroxy-4h-Pyrrolo[3,2,1-De][1,5]naphthyridin-7(5h)-One |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
(3S)-3-[[4-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethylamino)piperidin-1-yl]methyl]-5,10-difluoro-3-hydroxy-1,7-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7,9-tetraen-11-one |
NA |
289000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |