| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
(2S)-6-[(3R)-3-(1-aminocyclopropyl)pyrrolidin-1-yl]-8-fluoro-2-methyl-12-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,10-tetraene-11-carboxylic acid |
NA |
126000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
(2S)-6-[(3R)-3-(1-aminocyclopropyl)pyrrolidin-1-yl]-8-chloro-7-fluoro-2-methyl-12-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),10-tetraene-11-carboxylic acid |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
(2S)-6-[(3R)-3-(1-aminocyclopropyl)pyrrolidin-1-yl]-7,8-difluoro-2-methyl-12-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),10-tetraene-11-carboxylic acid |
NA |
211000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Sildenafil |
NA |
158489 |
NA |
NA |
NA |
NA |
PubChem |
| KCNH2 |
Vardenafil |
NA |
316228 |
NA |
NA |
NA |
NA |
PubChem |
| KCNH2 |
clozapine N-oxide |
NA |
133299.95 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
Eltrombopag |
NA |
1584890 |
NA |
NA |
NA |
NA |
PubChem |
| KCNH2 |
methyl (4aS,6aR,6bS,8aR,12R,12aS,14aR,14bS)-10-[[4-[[(4S)-4-amino-5-methoxy-5-oxopentanoyl]amino]phenyl]methoxy]-11-cyano-12-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-14-oxo-3,4,5,6,7,8,8a,12,14a,14b-decahydro-1H-picene-4a-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
(3R,4R)-4-[(3S)-3-(3-fluoro-6-methoxyquinolin-4-yl)-3-hydroxypropyl]-1-[3-(1,2-oxazol-5-yl)cyclobutyl]piperidine-3-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
1,3-dimethyl-5-[[4-[4-(trifluoromethyl)phenyl]-4H-pyrazol-1-ium-1-yl]methyl]pyrazole |
NA |
137000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3-[4-[(3-chlorobenzoyl)amino]phenyl]-N-(4-fluorophenyl)oxetane-3-carboxamide |
NA |
9094000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3,3-difluoro-N-(4-fluorophenyl)-1-[4-[4-(hydroxymethyl)-6-(trifluoromethyl)pyridin-3-yl]phenyl]cyclobutane-1-carboxamide |
NA |
6096000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3-[4-(6-cyclopropylpyridin-3-yl)phenyl]-N-(4-fluorophenyl)oxetane-3-carboxamide |
NA |
13450000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Ido1-IN-18 |
NA |
22840000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
N-(4-fluorophenyl)-1-[4-[4-(hydroxymethyl)-6-(trifluoromethyl)pyridin-3-yl]phenyl]cyclobutane-1-carboxamide |
NA |
11910000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Ido1-IN-19 |
NA |
21310000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3-[4-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)phenyl]-N-(4-fluorophenyl)oxetane-3-carboxamide |
NA |
13830000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3-[4-(6-cyclopropyl-4-methylpyridin-3-yl)phenyl]-N-(4-fluorophenyl)oxetane-3-carboxamide |
NA |
15890000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
N-(4-fluorophenyl)-3-[4-[4-methyl-6-(trifluoromethyl)pyridin-3-yl]phenyl]oxetane-3-carboxamide |
NA |
2228000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
2-[ethyl-[2-[(2S)-2-[4-[(5-fluoro-1,3-thiazol-2-yl)carbamoyl]-5-methylthiophen-2-yl]pyrrolidin-1-yl]-2-oxoethyl]amino]acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |