| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
(R)-2-(4-(((S)-3-((R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl)thiazolidine-2-carboxamido)methyl)phenylamino)-3-methylbutanoic acid hydrochloride |
NA |
NA |
NA |
408000 |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
(3R)-3-[[4-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethylamino)piperidin-1-yl]methyl]-5-fluoro-1,7-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7,9-tetraen-11-one |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
6-cyano-N-[(1R)-1-[1-ethyl-6-(trifluoromethyl)imidazo[4,5-c]pyridin-2-yl]ethyl]pyridine-3-sulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
6-cyano-N-[(1R)-1-(6-cyclopropyl-1-ethylimidazo[4,5-c]pyridin-2-yl)ethyl]pyridine-3-sulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
1-[2-[(3S,4S)-4-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethylamino)-3-methoxypiperidin-1-yl]ethyl]-2-oxoquinoline-7-carbonitrile |
NA |
176000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
1-[2-[(3R,4S)-3-hydroxy-4-[(3-oxo-4H-pyrido[3,2-b][1,4]oxazin-6-yl)methylamino]piperidin-1-yl]ethyl]-2-oxoquinoline-7-carbonitrile |
NA |
305000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
6-[[[(3R,4S)-3-hydroxy-1-[2-(7-methoxy-2-oxoquinoxalin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one |
NA |
172000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
Azd-9742 |
NA |
233000|200000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
1-[2-[(3S,4R)-4-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethylamino)-3-methoxypiperidin-1-yl]ethyl]-2-oxoquinoline-7-carbonitrile |
NA |
174000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
1-[2-((3R,4R)-3-methoxy-4-{[(3-oxo-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-6-yl)methyl]amino}piperidin-1-yl)ethyl]-2-oxo-1,2-dihydroquinoline-7-carbonitrile |
NA |
124000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
Gepotidacin |
NA |
1310000|1400000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| KCNH2 |
|
NA |
1584893 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Carbamazepine |
NA |
104712.85|104713 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Cetirizine |
NA |
108000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| KCNH2 |
Ciprofloxacin |
NA |
954992.59|954993|966000|NA |
NA |
NA |
NA |
NA|350002 |
BindingDB|PubChem |
| KCNH2 |
|
NA |
133300 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Maraviroc |
NA |
125893 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| KCNH2 |
(-)-(S)-9-Fluoro-2,3-dihydro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-7H-pyrido(1,2,3-de)-1,4-benzoxazine-6-carboxylic acid, hemihydrate |
NA|150000 |
912011|NA|915000|5000000|2300000|2100000|1100000 |
NA |
NA |
NA |
NA|739997 |
PubChem |
| KCNH2 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| KCNH2 |
Lidocaine |
NA |
263026.8|263027 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |