| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
7-((R)-3-((S)-1-(2-cyanoethylamino)ethyl)pyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-8-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
7-((R)-3-((S)-1-amino-2-cyanoethyl)pyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-8-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
7-((R)-3-((S)-1-amino-2-cyanoethyl)pyrrolidin-1-yl)-1-cyclopropyl-8-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
6-[(3R)-3-[(1S)-1-(2-cyanoethylamino)ethyl]pyrrolidin-1-yl]-7-fluoro-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxylic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
6-[(3R)-3-[(1S)-1-amino-2-cyanoethyl]pyrrolidin-1-yl]-7-fluoro-2-methyl-10-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,11-tetraene-11-carboxylic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
7-(3-(Aminomethyl)-3-methylazetidin-1-yl)-1-cyclopropyl-6-fluoro-8-methyl-4-oxo-1,4-dihydroquinoline-3-carboxylic acid |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
7-(3-((2-Cyanoethylamino)methyl)-3-methylazetidin-1-yl)-1-cyclopropyl-6-fluoro-8-methyl-4-oxo-1,4-dihydroquinoline-3-carboxylic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
(S)-1-((3R,4R)-1-(4-(5-methyl-1,3,4-oxadiazol-2-yl)benzyl)-3-aminopyrrolidine-4-carbonyl)pyrrolidine-2-carbonitrile |
NA |
165000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
(3R,4R)-4-amino-3-(pyrrolidine-1-carbonyl)-1-(quinoxaline-3-carbonyl)pyrrolidin-2-one |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
N-(3-methylphenyl)-2-pyridin-3-yl-1,3-thiazole-4-carboxamide |
NA |
279000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
2-[4-[[4-[3-Chloro-4-(hydroxymethyl)phenoxy]piperidin-1-yl]methyl]piperidine-1-carbonyl]-4-methylbenzoic acid |
NA |
100000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
Methyl 4-[4-[[4-[3-chloro-4-(hydroxymethyl)phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]butanoate |
NA |
20417379|20417379.45 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
[9-[[2-(2-methoxyphenoxy)phenyl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-[2-(2H-tetrazol-5-yl)phenyl]methanone |
NA |
512861384 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
[2-Chloro-4-[1-(piperidin-4-ylmethyl)piperidin-4-yl]oxyphenyl]methanol |
NA |
2951209|2951209.23 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
2-[4-[[4-[3-Chloro-4-(hydroxymethyl)phenoxy]piperidin-1-yl]methyl]piperidine-1-carbonyl]benzoic acid |
NA |
97723722|97723722.1 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
2-[4-[[4-[3-Chloro-4-(hydroxymethyl)phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]-3-(4-methylsulfonylphenyl)propanoic acid |
NA |
85113804|85113803.82 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
2-[4-[[4-[3-Chloro-4-(hydroxymethyl)phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]benzoic acid |
NA |
645654229 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
6-[4-[[4-[3-Chloro-4-(hydroxymethyl)phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxylic acid |
NA |
66069345|66069344.8 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
2-[4-[[4-[3-Chloro-4-(hydroxymethyl)phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]acetic acid |
NA |
64565423|64565422.9 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
3-[4-[[4-[3-Chloro-4-(hydroxymethyl)phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]benzoic acid |
NA |
512861384 |
NA |
NA |
NA |
NA |
BindingDB|TTD |