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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KCNH2 Indomethacin NA 301995.17|301995 NA NA NA NA BindingDB|PubChem|TTD
KCNH2 Irbesartan NA 194984.46|194984 NA NA NA NA BindingDB|PubChem|TTD
KCNH2 Lamotrigine NA 229086.77|251189|398107|229087|251188.64 NA NA NA NA BindingDB|PubChem|TTD
KCNH2 Lomefloxacin NA 2398832.92|2398830 NA NA NA NA BindingDB|PubChem|TTD
KCNH2 Bardoxolone Methyl NA 200000 NA NA NA NA PubChem|TTD
KCNH2 Mepivacaine NA 154881.66|154882 NA NA NA NA BindingDB|PubChem|TTD
KCNH2 Sitagliptin NA 158489|501187|1000000|501187.23 NA NA NA NA BindingDB|PubChem|TTD
KCNH2 5-Chloro-2-[(5-chloro-1,3-benzoxazol-2-yl)amino]benzoic acid NA NA NA 107200 NA NA BindingDB
KCNH2 3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid NA 3981071.71 NA NA NA NA BindingDB
KCNH2 5-Chloro-3-ethyl-1-(4-fluorophenyl)-1H-indole NA 3467368.5 NA NA NA NA BindingDB|TTD
KCNH2 1-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-yl]-propan-1-ol NA 2187761.62 NA NA NA NA BindingDB
KCNH2 5-Chloro-1-(4-fluoro-phenyl)-3-propyl-1H-indole NA 25703957.83 NA NA NA NA BindingDB
KCNH2 1-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-yl]-propan-1-one NA 1995262.31 NA NA NA NA BindingDB
KCNH2 1-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-yl]-ethanol NA 4570881.9 NA NA NA NA BindingDB|TTD
KCNH2 5-Chloro-3-(1-ethyl-propyl)-1-(4-fluoro-phenyl)-1H-indole NA 1479108.39 NA NA NA NA BindingDB
KCNH2 4-(4-Fluoro-phenyl)-8-(2-hydroxy-2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one NA 24000000 NA NA NA NA TTD
KCNH2 Tert-butyl 1-(1-isopropylpiperazine-4-carbonyl)piperidine-4-carboxylate NA 101111.1111|101111.11 NA NA NA NA BindingDB|TTD
KCNH2 (3,4-dihydroisoquinolin-2(1H)-yl)(4-isopropylpiperazin-1-yl)methanone NA 115000 NA NA NA NA BindingDB|TTD
KCNH2 (6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)(4-isopropylpiperazin-1-yl)methanone NA 115000 NA NA NA NA BindingDB|TTD
KCNH2 7-[(3S)-3-[(2-cyanoethylamino)methyl]pyrrolidin-1-yl]-1-cyclopropyl-6-fluoro-8-methoxy-4-oxoquinoline-3-carboxylic acid 106000 NA NA NA NA NA BindingDB|TTD