| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
Ofloxacin |
NA |
1412537.54|1412538|1420000|1412540|NA |
NA |
NA |
NA |
NA|470002 |
BindingDB|PubChem|TTD |
| KCNH2 |
6-((((1R,4r)-4-((R)-1-Amino-2-(7-methoxy-2-oxo-1,5-naphthyridin-1(2H)-yl)ethyl)cyclohexyl)amino)methyl)-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-one |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
6-[[[4-[(1R)-1-amino-2-(7-methoxy-2-oxoquinoxalin-1-yl)ethyl]cyclohexyl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
2-[[[4-[(1R)-1-amino-2-(7-methoxy-2-oxoquinoxalin-1-yl)ethyl]cyclohexyl]amino]methyl]-8H-pyrimido[5,4-b][1,4]oxazin-7-one |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
6-[[[4-[(1R)-1-amino-2-(7-fluoro-2-oxoquinoxalin-1-yl)ethyl]cyclohexyl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one |
NA |
174000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
2-[[[4-[(1R)-1-amino-2-(7-fluoro-2-oxoquinoxalin-1-yl)ethyl]cyclohexyl]amino]methyl]-8H-pyrimido[5,4-b][1,4]oxazin-7-one |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
6-[[[4-[(1R)-1-amino-2-(7-fluoro-4-methyl-2-oxoquinolin-1-yl)ethyl]cyclohexyl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one |
NA |
333000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
N2-(benzo[d][1,3]dioxol-5-ylmethyl)-N4-(pyridin-4-yl)-6-(trifluoromethyl)pyrimidine-2,4-diamine |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
(R)-2-methyl-6-(2-(2-methylpyrrolidin-1-yl)ethyl)quinoline |
NA |
216000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
4-[6-(azetidine-1-carbonyl)-5-fluoropyridin-3-yl]oxy-2-ethyl-N-(5-methylpyrazin-2-yl)indazole-6-carboxamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
5-[(2r,4s)-2-(Phenylmethyl)piperidin-4-Yl]-1,2-Oxazol-3-One |
NA |
1000000000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
5-[(2S,4S)-2-(2-phenylethyl)piperidin-4-yl]-1,2-oxazol-3-one |
NA |
1000000000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
5-[(2R,4S)-2-(2,2-Dimethylpropyl)-4-piperidinyl]-3(2H)-isoxazolone |
NA |
1000000000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
Pentobarbital |
NA |
131825.67|22800000|131826 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Phenobarbital |
NA |
3000000|3019951.72|3019950 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Procainamide |
NA |
138038.43|138038 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Pritelivir |
NA |
160000 |
NA |
NA |
NA |
NA |
PubChem |
| KCNH2 |
5-amino-1-(2-fluorophenyl)-N-(5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl)-1H-pyrazole-4-carboxamide |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
|
NA |
158489 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Rhynchophylline |
NA |
773000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |