| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
Codeine |
NA |
301995.17|301995 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Morphine |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Pf-05175157 |
NA |
141000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
[(2S,3S,4R,6S)-6-[(2R,3S,4R,5R,6S)-6-[[(4R,5S,6S,7R,9R,10R,11Z,13E,16R)-4-acetyloxy-10-hydroxy-5-methoxy-9,16-dimethyl-2-oxo-7-(2-oxoethyl)-1-oxacyclohexadeca-11,13-dien-6-yl]oxy]-4-(dimethylamino)-5-hydroxy-2-methyloxan-3-yl]oxy-4-hydroxy-2,4-dimethyloxan-3-yl] 3-methylbutanoate |
NA |
102329.3 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
N-ethyl-2-[3-(trifluoromethyl)phenyl]ethanamine |
NA |
537031.8 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
1-cyclopropyl-6-fluoro-7-[(8Z)-8-methoxyimino-2,6-diazaspiro[3.4]octan-6-yl]-4-oxo-2,3-dihydro-1,8-naphthyridine-3-carboxylic acid |
NA |
218776.16 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
Gatifloxacin |
NA |
128824.96|128825|130000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
2,6-Dimethyl-4-(2-nitrophenyl)-3,4-dihydropyridine-3,5-dicarboxylic acid dimethyl ester |
NA |
275000|280000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
[(1S,3R)-3-[[(3S,4S)-3-methoxyoxan-4-yl]amino]-1-propan-2-ylcyclopentyl]-[4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]piperazin-1-yl]methanone |
NA |
3900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
2-[(4-{2-[3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl}-4-phenylpiperidin-1-yl)carbonyl]benzoic acid |
NA |
125892.54 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
Raltegravir |
NA |
316228|1584893|3162278|3162280|1584890 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| KCNH2 |
imino-methyl-[1-[6-[(3R)-3-methylmorpholin-4-yl]-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrimidin-4-yl]cyclopropyl]-oxo-lambda6-sulfane |
NA |
166000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| KCNH2 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| KCNH2 |
Alvimopan |
NA |
794328|63095734|63095700|63095734.45 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Trimethoprim |
NA |
239883|239883.29 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
8-[2-[4-(2,3-Dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethylamino)piperidin-1-yl]ethyl]-2-methoxypyrido[2,3-d]pyrimidin-7-one |
NA |
206000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
2-(trans-4-(4-(7-Aminopyrazolo[1,5-a]pyrimidin-6-yl)phenyl)cyclohexyl)acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
2-(4-(Cyclohexylmethyl)piperazin-1-yl)-8-nitro-6-(trifluoromethyl)-4H-benzo(e)(1,3)thiazin-4-one |
NA |
101700 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
2-[[2-[(3R)-3-aminopiperidin-1-yl]-6-methyl-4-oxo-7H-pyrrolo[2,3-d]pyrimidin-3-yl]methyl]benzonitrile |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |