| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
Everolimus |
NA |
501187|794328|15848932|15848900|15848931.92 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Bupivacaine Hydrochloride |
NA |
866000|265000 |
NA |
NA |
NA |
NA |
PubChem |
| KCNH2 |
N-(1-(Piperidin-4-yl)indolin-5-yl)thiophene-2-carboximidamide dihydrochloride |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Ambrisentan |
NA |
501187|7943282|7943280|501187.23 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Premafloxacin |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
2-[1-[2-fluoro-4-[(5R)-2-oxo-5-(triazol-1-ylmethyl)-1,3-oxazolidin-3-yl]phenyl]piperidin-4-ylidene]propanenitrile |
NA |
213320 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
Grepafloxacin |
NA |
104000|NA |
NA |
NA |
NA |
NA|1000000 |
BindingDB|PubChem |
| KCNH2 |
Doripenem |
NA |
5011872|7943282|7943280|5011870|5011872.34 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
Kv1.5-IN-IIII |
NA |
418350 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
(3S)-3-[[4-(2,3-dihydro-[1,4]dioxino[2,3-c]pyridin-7-ylmethylamino)piperidin-1-yl]methyl]-5-fluoro-3-hydroxy-1,9-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12),9-tetraen-11-one |
NA |
101000|206000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
(2S,4S)-1-[(2S)-2-amino-3-(1,3-thiazol-4-yl)propanoyl]-4-fluoropyrrolidine-2-carbonitrile |
NA |
176600 |
NA |
NA |
NA |
NA |
TTD |
| KCNH2 |
(S)-5-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,4-triazole-3-carboxamide |
NA |
195000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
(10S)-4-(1H-indol-4-yl)-6-(4-methylsulfonyloxan-4-yl)-8,12-dioxa-1,3,5-triazatricyclo[8.4.0.02,7]tetradeca-2,4,6-triene |
NA |
6000000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
(9S)-9-Amino-9-deoxyerythromycin |
NA |
316227.77 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
N-methyl-1-[(10S)-6-(2-methylsulfonylpropan-2-yl)-8,12-dioxa-1,3,5-triazatricyclo[8.4.0.02,7]tetradeca-2,4,6-trien-4-yl]benzimidazol-2-amine |
NA |
4000000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Miristalkonium chloride |
NA |
NA |
NA |
NA |
1000000 |
NA |
PubChem |
| KCNH2 |
6-{4-[4-(4-Fluoro-3-trifluoromethyl-phenyl)-1-methyl-1H-imidazol-2-yl]-piperidin-1-yl}-5-methoxy-pyrimidin-4-ylamine |
NA |
670000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
Nicotine |
NA |
244300|245470.89|245471 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNH2 |
5-[[[(3S,4R)-3-fluoro-1-[2-(7-fluoro-2-oxo-1,5-naphthyridin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-2-methylpyridine-3-carbonitrile |
NA |
133000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNH2 |
5-[[[(3S,4R)-3-methoxy-1-[2-(7-methoxy-2-oxo-1,5-naphthyridin-1-yl)ethyl]piperidin-4-yl]amino]methyl]-2-methylpyridine-3-carbonitrile |
NA |
151000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |