| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KCNH2 |
(4r)-3-Fluoro-4-Hydroxy-4-{[(1r,4r)-4-{[(3-Oxo-3,4-Dihydro-2h-Pyrido[3,2-B][1,4]oxazin-6-Yl)methyl]amino}-2-Oxabicyclo[2.2.2]oct-1-Yl]methyl}-4,5-Dihydro-7h-Pyrrolo[3,2,1-De][1,5]naphthyridin-7-One |
NA |
174000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNH2 |
3-(1-Methylpyrrolidin-2-yl)pyridine |
NA |
245470.89|245471 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNJ1 |
3-[1-[(2R)-2-hydroxy-2-(4-methyl-1-oxo-3H-2-benzofuran-5-yl)ethyl]piperidin-4-yl]-1-(4-methyl-5-oxo-2H-furan-3-yl)pyrrolidin-2-one |
NA |
7000000 |
NA |
NA |
NA |
NA |
BindingDB |
| KCNJ11 |
2-Methyl-N-[2-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-naphthalen-1-yl]-butyramide |
NA |
NA |
NA |
177000 |
NA |
NA |
TTD |
| KCNJ11 |
Tifenazoxide |
NA |
696000|685000|165000 |
NA |
NA |
NA |
NA |
PubChem |
| KCNJ11 |
Diazoxide |
NA |
198000|194000|750000|740000 |
NA |
NA |
NA |
NA |
PubChem |
| KCNK18 |
Flufenamic Acid |
NA |
NA |
NA |
474000 |
NA |
NA |
PubChem |
| KCNK2 |
Lidocaine |
NA |
207000|180000 |
NA |
NA |
NA |
NA |
PubChem |
| KCNK2 |
Mexiletine |
NA |
173000 |
NA |
NA |
NA |
NA |
PubChem |
| KCNK2 |
Riluzole |
NA |
NA |
NA |
139400 |
NA |
NA |
PubChem |
| KCNK3 |
Lidocaine |
NA |
222000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| KCNK3 |
Mepivacaine |
NA |
709000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| KCNK3 |
Tetracaine |
NA |
668000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| KCNK9 |
Ethyl 2-(3-aminophenyl)-8,9-dimethoxy-3-methyl-5,6-dihydropyrrolo[2,1-a]isoquinoline-1-carboxylate |
NA |
268100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNK9 |
8,9-Dimethoxy-3-methyl-2-phenyl-5,6-dihydropyrrolo[2,1-a]isoquinoline-1-carbonitrile |
NA |
189200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNK9 |
Mevastatin |
NA |
159000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KCNMA1 |
5-(benzotriazol-1-yl)-2H-triazole-4-carboxamide |
NA |
112201.85 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNMA1 |
5-(5-methoxybenzotriazol-1-yl)-2H-triazole-4-carboxamide |
NA |
154881.66 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNMA1 |
5-(2-nitroanilino)-2H-triazole-4-carboxamide |
NA |
104712.85 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KCNN1 |
1-Ethyl-2-benzimidazolinone |
NA |
NA |
NA |
650000 |
NA |
NA |
BindingDB |