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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KCNQ1 Ambrisentan NA 501187 NA NA NA NA PubChem
KCNQ1 Dofetilide NA 251189|158489 NA NA NA NA PubChem
KCNQ1 Doripenem NA 316228 NA NA NA NA PubChem
KDM1A US10519118, Example 145 NA 114000 NA NA NA NA BindingDB
KDM1A 4-(4-Methoxyanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-Phenyl-2-prop-2-ynylsulfanyl-6-[3-(trifluoromethyl)anilino]pyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-(2-Chloroanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-(4-Chloroanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 125000|125026 NA NA NA NA BindingDB|TTD
KDM1A 4-(3-Chloroanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-(4-Fluoroanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 125000|125026 NA NA NA NA BindingDB|TTD
KDM1A 4-(4-Nitroanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 123310|124671 NA NA NA NA BindingDB|TTD
KDM1A 4-(4-Methylanilino)-6-phenyl-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-(4-Chlorophenyl)-6-(4-methoxyanilino)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-(4-Chlorophenyl)-2-prop-2-ynylsulfanyl-6-[3-(trifluoromethyl)anilino]pyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-(4-Bromophenyl)-6-(4-chloroanilino)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-(4-Methoxyanilino)-2-prop-2-ynylsulfanyl-6-(3,4,5-trimethoxyphenyl)pyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 2-Prop-2-ynylsulfanyl-4-[3-(trifluoromethyl)anilino]-6-(3,4,5-trimethoxyphenyl)pyrimidine-5-carbonitrile NA 125000 NA NA NA NA TTD
KDM1A 4-Chloro-6-(4-chlorophenyl)-2-[[1-[(2-chlorophenyl)methyl]triazol-4-yl]methylsulfanyl]pyrimidine-5-carbonitrile NA 125000|125026 NA NA NA NA BindingDB|TTD
KDM1A [[5-Cyano-2-[(4-fluorophenyl)methylsulfanyl]-6-(3,4,5-trimethoxyphenyl)pyrimidin-4-yl]amino]thiourea NA 125000|125026 NA NA NA NA BindingDB|TTD
KDM1A US10519118, Example 132 NA 173000 NA NA NA NA BindingDB