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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KDM1A (2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-carbamimidamido-2-[[(2S)-2-[(2-hydroxyacetyl)amino]propanoyl]amino]pentanoyl]amino]-3-hydroxybutanoyl]amino]-4-methylsulfanylbutanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[(2-hydroxyacetyl)amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-N-[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]pentanediamide 500000 NA NA NA NA NA TTD
KDM1A 2-(4-cyano-N-(4-methylphenyl)sulfonylanilino)-N-pyridin-3-ylacetamide NA 150000 NA NA NA NA TTD
KDM1A deamino-Gly(OH)-Ala-Arg-Thr-Met-Gln-Thr-Ala-Arg-Lys-Ser-Thr-Gly-Gly-Lys-Ala-Pro-Arg-Lys-Gln-Leu-NH2 500000 NA NA NA NA NA TTD
KDM1A H-Arg-Thr-Met-Gln-Thr-Ala-Arg-Lys-Ser-Thr-Gly-Gly-Lys-Ala-Pro-Arg-Lys-Gln-Leu-NH2 500000 NA NA NA NA NA TTD
KDM1A 4-[[5-Chloro-1-[(4-fluorophenyl)methyl]indol-3-yl]-hydroxymethyl]-3-methylideneoxolan-2-one NA NA 202000 NA NA NA BindingDB
KDM1A H-Ala-Arg-Thr-Met-Gln-Thr-Ala-Arg-Lys-Ser-Thr-OH NA NA 140000 NA NA NA BindingDB
KDM1A Tranylcypromine NA|242000|243000|357000|284000 NA 101000|NA NA NA NA BindingDB|PubChem
KDM1A N-(4-acetyl-1,3-thiazol-2-yl)benzamide NA 188000 NA NA NA NA TTD
KDM1A (+)-Tranylcypromine 168000|243000|284000 NA NA NA NA NA BindingDB|PubChem
KDM1A 1-[2-(4-Chloroanilino)-1,3-thiazol-4-yl]ethanone NA 121000|249000 NA NA NA NA ChEMBL|TTD
KDM1A 1-[2-(2-Chloroanilino)thiazole-4-yl]ethanone NA 437000|188000 NA NA NA NA ChEMBL|TTD
KDM1A 2-(4-Methoxyphenyl)Cyclopropanamine 188000 NA NA NA NA NA BindingDB|TTD
KDM1A 1-(6-Bromonaphthalen-2-yl)oxy-3-(cyclopropylamino)propan-2-ol NA 111400 NA NA NA NA BindingDB|TTD
KDM1A 6-(5,6-dimethoxybenzimidazol-1-yl)-N-piperidin-4-ylpyridin-2-amine 170000 NA NA NA NA NA BindingDB
KDM1A Jhdm-IN-1 NA 620000 NA NA NA NA TTD
KDM1A Parnate NA|243000 184000|242000|NA NA NA NA NA BindingDB|PubChem
KDM1A N-(4-acetyl-1,3-thiazol-2-yl)benzenesulfonamide NA 188000 NA NA NA NA TTD
KDM1A 1-(4-Acetyl-1,3-thiazol-2-yl)-3-phenylurea NA 188000 NA NA NA NA TTD
KDM1A Gsk2879552 NA 403900 NA NA NA NA BindingDB|PubChem
KDM1A N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]benzamide NA 188000 NA NA NA NA TTD