Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KDM1A Tert-butyl 4-[[1-[2-(4-fluorophenyl)ethyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[2-(2-oxochromen-4-yl)oxyethyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-(naphthalen-2-ylmethyl)triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A tert-butyl 4-[[1-[(2-oxo-1H-quinolin-4-yl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A tert-butyl 4-[[1-(1H-benzimidazol-2-ylmethyl)triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A tert-butyl 4-[[1-[(5-oxo-2H-furan-3-yl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-(2-oxochromen-4-yl)triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Fluorophenyl)methyl]triazol-4-yl]methyl 4-methylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Methylphenyl)methyl]triazol-4-yl]methyl 4-methylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Fluorophenyl)methyl]triazol-4-yl]methyl 4-methylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Chlorophenyl)methyl]triazol-4-yl]methyl 4-methylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Methylphenyl)methyl]triazol-4-yl]methyl 4-ethylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Fluorophenyl)methyl]triazol-4-yl]methyl 4-ethylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Fluorophenyl)methyl]triazol-4-yl]methyl 4-(2-hydroxyethyl)piperazine-1-carbodithioate NA 100100 NA NA NA NA BindingDB|TTD
KDM1A [1-[(4-Fluorophenyl)methyl]triazol-4-yl]methyl 4-(2-hydroxyethyl)piperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Fluorophenyl)methyl]triazol-4-yl]methyl 4-phenylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Fluorophenyl)methyl]triazol-4-yl]methyl 4-phenylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Fluorophenyl)methyl]triazol-4-yl]methyl piperidine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Fluorophenyl)methyl]triazol-4-yl]methyl piperidine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Methylphenyl)methyl]triazol-4-yl]methyl piperidine-1-carbodithioate NA 125000 NA NA NA NA TTD