| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KDM1A |
1-[2-(4-Methoxyanilino)-1,3-thiazol-4-yl]ethanone |
NA |
188000 |
NA |
NA |
NA |
NA |
TTD |
| KDM1A |
2-[[5-Cyano-6-(4-nitrophenyl)-2-prop-2-ynylsulfanylpyrimidin-4-yl]amino]guanidine |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| KDM1A |
4-Chloro-6-(4-nitrophenyl)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile |
NA |
125000|125026|125025.9 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KDM1A |
4-Chloro-6-(3-chlorophenyl)-2-prop-2-ynylsulfanylpyrimidine-5-carbonitrile |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| KDM1A |
4-[2-(Piperidin-4-ylamino)cyclopropyl]phenol |
NA |
8776000 |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1A |
N-(4-(4-Chlorophenyl)-2-thiazolyl)-N'-phenylurea |
NA |
188000 |
NA |
NA |
NA |
NA |
TTD |
| KDM1B |
(1S,2R)-2-(4-bromo-3-fluorophenyl)cyclopropan-1-amine |
280000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-[3-fluoro-4-(trifluoromethyl)phenyl]cyclopropan-1-amine |
180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-(3,6-difluoro-2-phenylmethoxyphenyl)cyclopropan-1-amine |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-(4-bromo-5-fluoro-2-methylphenyl)cyclopropan-1-amine |
280000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-(4-bromo-2-fluoro-6-phenylmethoxyphenyl)cyclopropan-1-amine |
490000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-[4-bromo-2-(trifluoromethyl)phenyl]cyclopropan-1-amine |
390000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-(4-bromo-2,5-difluorophenyl)cyclopropan-1-amine |
180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1R,2R)-2-(2-fluoro-6-phenylmethoxyphenyl)cyclopropan-1-amine |
370000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1R,2R)-2-[4-bromo-2-(trifluoromethyl)phenyl]cyclopropan-1-amine |
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-(4-bromo-3,5-difluorophenyl)cyclopropan-1-amine |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-(2-fluoro-6-phenylmethoxyphenyl)cyclopropan-1-amine |
240000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
5-[(1R,2S)-2-aminocyclopropyl]-2-bromophenol |
290000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
Tranylcypromine |
186000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-(4-Bromophenyl)cyclopropan-1-amine |
740000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |