| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KDM4A |
3-[9-Cyclopentylnonanoyl(hydroxy)amino]propanoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
N-(9-Cyclopropyl-1-oxononyl)-N-hydroxy-beta-alanine |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
Methyl 3-[hydroxy(10-methylundecanoyl)amino]propanoate |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
Pyrazole |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
1H-Pyrazole-5-boronic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
2-(5-Amino-2-methoxyphenyl)pyridine-4-carboxylic acid |
NA |
310000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
1,5-Dimethyl-1H-pyrazole-4-carboxylic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
4-Bromo-1-methyl-2-phenyl-1H-imidazole |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
1-Benzyl-4-bromo-1h-1,2,3-triazole |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
1-Benzyl-4-bromo-3-oxidotriazol-3-ium |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
5-hydroxy-N,1-dimethyl-1H-1,2,3-triazole-4-carboxamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
4H-1,2,3-Triazole-4-thione, 2,3-dihydro-2,3,5-trimethyl- |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
1-methyl-1H-1,2,3-triazol-4-amine |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
(2S,3R)-3-[(dimethylamino)methyl]-1-phenylbicyclo[2.2.1]heptan-2-ol |
NA |
NA |
129000 |
NA |
NA |
NA |
ChEMBL |
| KDM4C |
(5-chloro-1-methyl-1H-imidazol-2-yl)methanol |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
4-Chloro(phenyl)thiazole |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
Daminozide |
NA |
2500000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
2-Methyl-2-[(propylcarbamoyl)amino]propanoic acid |
NA |
126000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
2-[3-(4-Methylpiperazine-1-carbonyl)pyrazol-1-yl]acetic acid |
NA |
387000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
1-methyl-1H-1,2,3-triazole-4-carboxylic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |