| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KDM1B |
Parnate |
NA |
2300000 |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1S,2R)-2-phenylcyclopropan-1-amine;(1R,2S)-2-phenylcyclopropan-1-amine |
NA |
2300000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| KDM1B |
N-((2S)-1-(Benzylamino)-1-oxo-6-((2-phenylcyclopropyl)amino)hexan-2-yl)-[1,1'-biphenyl]-4-carboxamide |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KDM1B |
N-[(2S)-1-oxo-6-[(2-phenylcyclopropyl)amino]-1-[[3-(trifluoromethyl)phenyl]methylamino]hexan-2-yl]-4-phenylbenzamide |
NA |
540000 |
NA |
NA |
NA |
NA |
TTD |
| KDM1B |
N-[(2S)-1-[(4-chlorophenyl)methylamino]-1-oxo-6-[(2-phenylcyclopropyl)amino]hexan-2-yl]-4-phenylbenzamide |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KDM1B |
(1S,2R)-2-(4-bromo-2-fluorophenyl)cyclopropan-1-amine |
270000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM1B |
(1R,2R)-2-(4-ethoxy-3-fluorophenyl)cyclopropan-1-amine |
290000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| KDM2A |
(2R)-2-hydroxypentanedioic acid |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| KDM3A |
N-[(5-chloro-8-hydroxyquinolin-7-yl)-(3-methylthiophen-2-yl)methyl]benzamide |
NA |
191000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| KDM3A |
Oxalylglycine |
NA |
569000 |
NA |
NA |
NA |
NA |
BindingDB |
| KDM4A |
2-(2-Azanyl-1,3-Thiazol-4-Yl)pyridine-4-Carboxamide |
NA |
104200 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
N-[6-(4-acryloyl-1,4-diazepan-1-yl)-2-(pyridin-2-yl)pyrimidin-4-yl]-beta-alanine |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
3-[[6-(4-Ethenylsulfonyl-1,4-diazepan-1-yl)-2-pyridin-2-ylpyrimidin-4-yl]amino]propanoic acid |
NA |
290000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
(2S,3R)-3-[(dimethylamino)methyl]-1-phenylbicyclo[2.2.1]heptan-2-ol |
170000|NA |
NA |
NA |
NA|105000 |
NA |
NA |
ChEMBL|TTD |
| KDM4A |
(2R,3S)-3-[(dimethylamino)methyl]-1-phenylbicyclo[2.2.1]heptan-2-ol |
NA |
NA |
NA |
1216000 |
NA |
NA |
ChEMBL|TTD |
| KDM4A |
Daminozide |
NA |
3300000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
Oxalylglycine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
3-(N-Hydroxy-7-methyloctanamido)propanoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
3-[[2-Pyridin-2-Yl-6-(1,2,4,5-Tetrahydro-3-Benzazepin-3-Yl)pyrimidin-4-Yl]amino]propanoic Acid |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4A |
3-[9-Cyclohexylnonanoyl(hydroxy)amino]propanoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |