| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| KDM4C |
1-phenyl-1H-1,2,3-triazol-4-amine |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
1-(4-methylbenzyl)-1H-1,2,3-triazole-4-carboxylic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
(3R)-5-oxo-1-(1,3-thiazol-2-yl)pyrrolidine-3-carboxylic acid |
NA |
676000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
4-nitro-1-phenyl-1H-pyrazole |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
1-phenyl-1H-1,2,3-triazole-5-carboxylic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
Oxalylglycine |
NA |
430000 |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
methyl 1-benzyl-5-hydroxy-1H-1,2,3-triazole-4-carboxylate |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
2-(Quinoline-2-carbonylamino)acetic acid |
NA |
2810000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
Nitrazepam |
NA|200000 |
200000|NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| KDM4C |
Benzoic acid, 5-[[(ethylamino)thioxomethyl]amino]-2-hydroxy- |
NA |
165000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
2-(2-Acetylphenyl)isonicotinic acid |
NA |
507000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
2,4-Dihydroxythiazole |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
2-(5-Hydroxy-7-methyl-2-oxochromen-4-yl)acetic acid |
NA |
176000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
1-Phenyl-1H-1,2,3-triazole-4-carboxylic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
3-Benzyl-5-chloro-1,2,3-triazole-1-oxide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
2-[5-(phenoxymethyl)-1H-1,2,3,4-tetrazol-1-yl]acetic acid |
NA |
2320000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| KDM4C |
1H-Pyrazole-5-carboxylic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
1-Phenyl-3-benzoyl-4-hydroxy-5-methylpyrazole |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
4,5-Dibromo-1-oxido-3-phenyltriazol-1-ium |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| KDM4C |
2-[(2-Chloropyridin-3-yl)amino]pyridine-3-carbonitrile |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |