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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KDM4C 2-phenyl-2H-1,2,3-triazole-4-carboxylic acid 200000 NA NA NA NA NA TTD
KDM4C Pyrazole-3,5-dicarboxylic acid monohydrate 200000 NA NA NA NA NA TTD
KDM4C Ethyl 5-methyl-1H-1,2,3-triazole-4-carboxylate 200000 NA NA NA NA NA TTD
KDM4C (2R)-2-[(4-chloropyridine-2-carbonyl)amino]propanoic acid NA 1210000 NA NA NA NA ChEMBL|TTD
KDM4C 5-Nitro-1H-pyrazole-3-carboxylic acid 200000 NA NA NA NA NA TTD
KDM4E 2,4-Pyridinedicarboxylic acid 914000 NA NA NA NA NA BindingDB
KDM4E Dipicolinic Acid NA 120000|250000 NA NA NA NA BindingDB
KDM4E Quinolinic Acid NA 10000000 NA NA NA NA PubChem
KDM4E Succinic Acid NA 710000 NA NA NA NA BindingDB
KDM4E 5-methyl-4-prop-2-enyl-2-pyridin-2-yl-1H-pyrazol-3-one NA 191000 NA NA NA NA BindingDB
KDM4E 3-[2-(1H-benzimidazol-2-yl)-5-methyl-3-oxo-1H-pyrazol-4-yl]propanoic acid NA 274000 NA NA NA NA BindingDB
KDM4E 2-[2-(1H-benzimidazol-2-yl)-3-oxo-1H-pyrazol-5-yl]acetic acid NA 347000 NA NA NA NA BindingDB
KDM4E methyl 3-[2-(1H-benzimidazol-2-yl)-4-methyl-3-oxo-1H-pyrazol-5-yl]propanoate NA 106000 NA NA NA NA BindingDB
KDM4E 3-[2-(1H-benzimidazol-2-yl)-4-methyl-3-oxo-1H-pyrazol-5-yl]propanoic acid NA 437000 NA NA NA NA BindingDB
KDM4E N,5-dihydroxy-2-methoxybenzamide NA 230000 NA NA NA NA BindingDB
KDM4E N,5-dihydroxy-2-phenoxybenzamide NA 360000 NA NA NA NA BindingDB
KDM4E 2-(1H-Benzoimidazol-2-yl)-5-methyl-2H-pyrazol-3-ylamine NA 199000 NA NA NA NA BindingDB
KDM4E Fumaric Acid NA 1600000 NA NA NA NA BindingDB
KDM4E (2S)-3-benzylsulfanyl-2-(oxaloamino)propanoic acid NA 200000 NA NA NA NA BindingDB|TTD
KDM4E N-(Carboxycarbonyl)-D-phenylalanine NA 320000 NA NA NA NA BindingDB