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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KDM5A 3-[4-(2-Butyl-1-benzofuran-3-carbonyl)phenoxy]propyl-triethylazanium;iodide NA 314000 NA NA NA NA BindingDB|TTD
KDM5A 3-[4-[C-(1-benzofuran-3-yl)-N-methylcarbonimidoyl]phenoxy]propyl-trimethylazanium;iodide NA 1310000 NA NA NA NA BindingDB|TTD
KDM5A Daminozide NA 2200000 NA NA NA NA BindingDB|TTD
KDM5A Amiodarone NA 1000000 NA NA NA NA PubChem
KDM5A Oxalylglycine NA 250000|640000 NA NA NA NA BindingDB|TTD
KDM5A Histone H3 (1-21) NA 571000 NA NA NA NA BindingDB|TTD
KDM5A 3-[[2-Pyridin-2-Yl-6-(1,2,4,5-Tetrahydro-3-Benzazepin-3-Yl)pyrimidin-4-Yl]amino]propanoic Acid NA 110000 NA NA NA NA BindingDB|TTD
KDM5A 2-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-diiodophenoxy]ethyl-trimethylazanium NA 1658000 NA NA NA NA BindingDB
KDM5A 3-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-diiodophenoxy]propyl-trimethylazanium NA 562000 NA NA NA NA BindingDB
KDM5A Methyl 3-[hydroxy(10-methylundecanoyl)amino]propanoate NA 210000 NA NA NA NA BindingDB|TTD
KDM5A 3-[Hydroxy(10-methylundecanoyl)amino]propanoic acid NA 110000 NA NA NA NA BindingDB|TTD
KDM5A 2-(Oxaloamino)-2-oxoacetic acid NA 250000 NA NA NA NA BindingDB
KDM5B Succinic Acid NA 1400000 NA NA NA NA BindingDB|PubChem
KDM5B Oxalylglycine NA 920000 NA NA NA NA BindingDB
KDM5B Citric Acid NA 800000 NA NA NA NA PubChem
KDM5B (2R)-2-hydroxypentanedioic acid NA|10000000 203000|NA|3600000 NA NA NA NA BindingDB|PubChem
KDM5B (2S)-2-hydroxypentanedioic acid NA 1600000 NA NA NA NA PubChem
KDM5B Alpha-Ketoglutaric Acid NA 800000 NA NA NA NA PubChem
KDM5B Oxaloacetic Acid NA 900000 NA NA NA NA PubChem
KDM5C 4HQ derivative 4 NA 443200 NA NA NA NA BindingDB