Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KDM5C methyl 4'-(phenethylcarbamoyl)-[2,2'-bipyridine]-4-carboxylate (N4) NA 450000 NA NA NA NA BindingDB
KDM5C N-[(5-chloro-8-hydroxyquinolin-7-yl)-(3-methylthiophen-2-yl)methyl]benzamide NA 178000 NA NA NA NA BindingDB|TTD
KDM5C NA 103400 NA NA NA NA BindingDB
KDM5C NA 111000 NA NA NA NA BindingDB
KDM5C 8-(1-methylpyrazol-3-yl)-3H-pyrido[3,4-d]pyrimidin-4-one NA 103400 NA NA NA NA TTD
KDM5C 8-(piperidin-1-ylmethyl)-3H-pyrido[3,4-d]pyrimidin-4-one NA 111000 NA NA NA NA TTD
KDM5C FG-2216 NA 549600 NA NA NA NA BindingDB
KDM5C 4HQ derivative 6 NA 159000 NA NA NA NA BindingDB
KDM5C 4HQ derivative 7 NA 465000 NA NA NA NA BindingDB
KDM5C 4HQ derivative 8 NA 122900 NA NA NA NA BindingDB
KDM6A Vorinostat NA 164000 NA NA NA NA BindingDB
KDM6B N-[(5-chloro-8-hydroxyquinolin-7-yl)-(3-methylthiophen-2-yl)methyl]benzamide NA 106000 NA NA NA NA TTD
KDM7A 3-[2-(2-Butyl-1-benzofuran-3-carbonyl)phenoxy]propyl-trimethylazanium;iodide NA 102000 NA NA NA NA BindingDB|TTD
KDM7A (2-Butyl-1-benzofuran-3-yl)-[4-[3-(dimethylamino)propoxy]phenyl]methanone NA 295000|333000 NA NA NA NA BindingDB|TTD
KDM7A Trimethyl-[3-[2-(2-methyl-1-benzofuran-3-carbonyl)phenoxy]propyl]azanium;iodide NA 326000 NA NA NA NA BindingDB|TTD
KDM7A [4-(3-Aminopropoxy)phenyl]-(2-butyl-1-benzofuran-3-yl)methanone NA 534000 NA NA NA NA BindingDB|TTD
KDM7A Trimethyl-[3-[4-(2-methyl-1-benzothiophene-3-carbonyl)phenoxy]propyl]azanium;iodide NA 104000 NA NA NA NA BindingDB|TTD
KDM7A 3-[4-(2-Butyl-1-benzofuran-3-carbonyl)phenoxy]propyl-triethylazanium;iodide NA 151000 NA NA NA NA BindingDB|TTD
KDM7A Amiodarone NA 156000 NA NA NA NA BindingDB|PubChem|TTD
KDM7A Oxalylglycine NA 250000 NA NA NA NA TTD