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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KDM7A 2-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-diiodophenoxy]ethyl-trimethylazanium;iodide NA 2232000 NA NA NA NA TTD
KDM7A 2-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-diiodophenoxy]ethyl-trimethylazanium NA 2232000 NA NA NA NA BindingDB
KDR N4-(3-bromo-4-fluorophenyl)-6-phenethyl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine NA 132100|198300 NA NA NA NA BindingDB|TTD
KDR Imipenem NA NA NA NA NA 300000 PubChem
KDR 5-[(1z)-2-(2-Methoxyphenyl)prop-1-En-1-Yl]furo[2,3-D]pyrimidine-2,4-Diamine NA 151900 NA NA NA NA BindingDB
KDR N-[5-[2-(cyclopropanecarbonylamino)imidazo[1,2-b]pyridazin-6-yl]oxy-2-methylphenyl]-2-(piperidin-1-ylmethyl)benzamide NA NA 110000 NA NA NA BindingDB
KDR N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[1-(cyclohexylamino)-2-methylsulfonylethyl]furan-2-yl]quinazolin-4-amine NA 200000 NA NA NA NA TTD
KDR N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[2-methylsulfonyl-1-(propan-2-ylamino)ethyl]furan-2-yl]quinazolin-4-amine NA 200000 NA NA NA NA TTD
KDR N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[2-methylsulfonyl-1-(2-methylsulfonylethylamino)ethyl]furan-2-yl]quinazolin-4-amine NA 200000 NA NA NA NA TTD
KDR [[(1S)-1-[5-[4-[3-chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]furan-2-yl]-2-methylsulfonylethyl]amino] propanoate NA 200000 NA NA NA NA TTD
KDR [[(1S)-1-[5-[4-[3-chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]furan-2-yl]-2-methylsulfonylethyl]amino] pentanoate NA 200000 NA NA NA NA TTD
KDR [[(1S)-1-[5-[4-[3-chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]furan-2-yl]-2-methylsulfonylethyl]amino] heptanoate NA 200000 NA NA NA NA TTD
KDR 2-(Dimethylamino)ethyl 4-methoxy-3-[[3-pyrimidin-5-yl-5-(trifluoromethyl)phenyl]carbamoylamino]benzoate NA 500000 NA NA NA NA TTD
KDR 2-(Diethylamino)ethyl 4-methoxy-3-[[5-pyrimidin-5-yl-2-(trifluoromethoxy)phenyl]carbamoylamino]benzoate NA 500000 NA NA NA NA TTD
KDR 2-[di(propan-2-yl)amino]ethyl 3-[[3-(1H-indol-5-yl)-5-(trifluoromethyl)phenyl]carbamoylamino]-4-methoxybenzoate NA 500000 NA NA NA NA TTD
KDR 2-[di(propan-2-yl)amino]ethyl 3-[[5-(1H-indol-5-yl)-2-(trifluoromethoxy)phenyl]carbamoylamino]-4-methoxybenzoate NA 500000 NA NA NA NA TTD
KDR 2-[Di(propan-2-yl)amino]ethyl 4-methoxy-3-[[5-pyrimidin-5-yl-2-(trifluoromethoxy)phenyl]carbamoylamino]benzoate NA 500000 NA NA NA NA TTD
KDR 2-[di(propan-2-yl)amino]ethyl 4-methoxy-3-[[5-(1H-pyrazol-4-yl)-2-(trifluoromethoxy)phenyl]carbamoylamino]benzoate NA 500000 NA NA NA NA TTD
KDR 2-[Di(propan-2-yl)amino]ethyl 4-methoxy-3-[[5-(1-methylpyrazol-4-yl)-2-(trifluoromethoxy)phenyl]carbamoylamino]benzoate NA 500000 NA NA NA NA TTD
KDR 2-Morpholin-4-ylethyl 4-methoxy-3-[[3-pyridin-3-yl-5-(trifluoromethyl)phenyl]carbamoylamino]benzoate NA 500000 NA NA NA NA TTD