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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KDM1A (1-Benzyltriazol-4-yl)methyl piperidine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Chlorophenyl)methyl]triazol-4-yl]methyl piperidine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A (1-Benzyltriazol-4-yl)methyl morpholine-4-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Fluorophenyl)methyl]triazol-4-yl]methyl morpholine-4-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Fluorophenyl)methyl]triazol-4-yl]methyl morpholine-4-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[(7-hydroxy-2-oxochromen-3-yl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 102560 NA NA NA NA TTD
KDM1A tert-butyl (2S)-2-benzamido-6-(prop-2-ynylamino)hexanoate NA 143600 NA NA NA NA BindingDB|TTD
KDM1A tert-butyl (2S)-2-benzamido-6-(but-2-ynylamino)hexanoate NA 131900 NA NA NA NA BindingDB|TTD
KDM1A N-[3-[3-(prop-2-ynylamino)propoxy]phenyl]benzamide NA 184200 NA NA NA NA BindingDB|TTD
KDM1A (1S,2R)-2-phenylcyclopropan-1-amine;(1R,2S)-2-phenylcyclopropan-1-amine NA|357000 242000|NA NA|101000 NA NA NA PubChem
KDM1A N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]methanesulfonamide NA 188000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[(6-methyl-2-oxochromen-4-yl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A 1-[2-(3-Hydroxyanilino)-1,3-thiazol-4-yl]ethanone NA 188000 NA NA NA NA TTD
KDM1A N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-N,4-dimethylbenzenesulfonamide NA 188000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[(7-hydroxy-5-methyl-2-oxochromen-4-yl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A 1-[2-(2-Methylanilino)-1,3-thiazol-4-yl]ethanone NA 188000 NA NA NA NA TTD
KDM1A 1-[2-(3-Chloroanilino)-1,3-thiazol-4-yl]ethanone NA 123000 NA NA NA NA ChEMBL|TTD
KDM1A N-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-1-phenylmethanesulfonamide NA 188000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[(2-oxochromen-3-yl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[(6-chloro-2-oxochromen-4-yl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD