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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
KDM1A Gsk-lsd1 NA NA 425000 NA NA NA BindingDB
KDM1A Tert-butyl 4-[[1-[[2-(trifluoromethyl)phenyl]methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Fluorophenyl)methyl]triazol-4-yl]methyl 4-benzylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Methylphenyl)methyl]triazol-4-yl]methyl 4-benzylpiperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-(2-fluorophenyl)triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2-Chlorophenyl)methyl]triazol-4-yl]methyl piperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Chlorophenyl)methyl]triazol-4-yl]methyl piperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(3,4-Dichlorophenyl)methyl]triazol-4-yl]methyl piperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(3,4,5-Trimethoxyphenyl)methyl]triazol-4-yl]methyl piperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A Benzyl 4-[[1-[(4-chlorophenyl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-(4-methylphenyl)triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[3-(trifluoromethyl)phenyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-(4-methoxyphenyl)triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A [1-[(2,6-Difluorophenyl)methyl]triazol-4-yl]methyl piperazine-1-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Methylphenyl)methyl]triazol-4-yl]methyl morpholine-4-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A [1-[(4-Chlorophenyl)methyl]triazol-4-yl]methyl morpholine-4-carbodithioate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[(2-methylphenyl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[[4-(trifluoromethyl)phenyl]methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[(4-nitrophenyl)methyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD
KDM1A Tert-butyl 4-[[1-[2-(4-methylphenyl)ethyl]triazol-4-yl]methylsulfanylcarbothioyl]piperazine-1-carboxylate NA 125000 NA NA NA NA TTD