Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| KCNA10 | Dalfampridine | NA | 1580000 | NA | NA | NA | NA | GtoPDB |
| KCNA2 | 9-Methoxyfuro[3,2-g][1,4]benzoxazin-3-one | NA | NA | 590000 | NA | NA | NA | BindingDB |
| KCNA3 | Dalfampridine | NA | NA | 195000 | NA | NA | NA | BindingDB|PubChem |
| KCNA3 | Bergapten | NA | 101000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| KCNA3 | Ethyl 1-(3-cyano-3,3-diphenylpropyl)piperidine-4-carboxylate | NA | 230000 | NA | NA | NA | NA | BindingDB|TTD |
| KCNA5 | Dalfampridine | NA | NA | 270000 | NA | NA | NA | GtoPDB |
| KCNA5 | Bergapten | NA | NA | 177000 | NA | NA | NA | PubChem |
| KCNA5 | Lidocaine | NA | 2188000 | NA | NA | NA | NA | PubChem|TTD |
| KCNA5 | Diltiazem | NA | NA | 115000 | NA | NA | NA | GtoPDB |
| KCNA5 | 6-((((1R,4r)-4-((R)-1-Amino-2-(7-methoxy-2-oxo-1,5-naphthyridin-1(2H)-yl)ethyl)cyclohexyl)amino)methyl)-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-one | NA | 333000 | NA | NA | NA | NA | TTD |
| KCNA5 | Methyl 2-[(4-butoxyphenyl)sulfonylamino]-3-phenylpropanoate | NA | 109740 | NA | NA | NA | NA | TTD |
| KCNA5 | 2-[3-[2-[(4-butoxyphenyl)sulfonylamino]ethyl]indol-1-yl]-N-(4-chlorophenyl)acetamide | NA | 185140 | NA | NA | NA | NA | TTD |
| KCNA6 | Bergapten | NA | NA | 187000 | NA | NA | NA | BindingDB|PubChem |
| KCNA6 | Tetraethylammonium | NA | 7000000 | NA | NA | NA | NA | GtoPDB |
| KCNB2 | Dalfampridine | NA | 1500000 | NA | NA | NA | NA | GtoPDB |
| KCNB2 | 2-(2-Aminoethyl)-5-methoxyindole | NA | 524000 | NA | NA | NA | NA | BindingDB |
| KCNB2 | Tetraethylammonium | NA | 2600000 | NA | NA | NA | NA | GtoPDB |
| KCNC1 | 5-Methoxymethyl-3-methyl-furo[3,2-g]chromen-7-one | NA | NA | 213000 | NA | NA | NA | BindingDB |
| KCNC1 | Bergapten | NA | NA | 111000 | NA | NA | NA | BindingDB|PubChem |
| KCNC1 | 5,8-Diethoxypsoralen | NA | NA | 178000 | NA | NA | NA | BindingDB |