Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| KAT7 | US11911372, Example 101 | NA | 107406 | NA | NA | NA | NA | BindingDB |
| KAT7 | 4-cyano-N-(5-phenylisoxazol-3-yl)benzenesulfonamide | NA | 123230 | NA | NA | NA | NA | BindingDB |
| KAT8 | 2-Hydroxy-5-pentadecylbenzoic acid | NA | 263026799190 | NA | NA | NA | NA | BindingDB |
| KAT8 | 2-Hydroxy-6-(11-hydroxyundecyl)benzoic acid | NA|157000 | 524807460250|NA | NA | NA | NA | NA | BindingDB |
| KAT8 | 5-Decyl-2-hydroxybenzoic acid | NA | 190546071796 | NA | NA | NA | NA | BindingDB |
| KAT8 | 4-Amino-3-methoxynaphthalen-1-ol | NA | 177000 | NA | NA | NA | NA | BindingDB |
| KAT8 | N-(4-hydroxynaphthalen-1-yl)decanamide | NA | 250000 | NA | NA | NA | NA | BindingDB |
| KAT8 | N-(4-hydroxynaphthalen-1-yl)-2-phenylacetamide | NA | 365000 | NA | NA | NA | NA | BindingDB |
| KAT8 | Anacardic Acid | NA | 213796208950 | NA | NA | NA | NA | BindingDB |
| KAT8 | 4-Methoxyphenylhydrazine hydrochloride | NA | 680000 | NA | NA | NA | NA | BindingDB |
| KAT8 | 4-Nitro-1-naphthol | NA | 141000 | NA | NA | NA | NA | BindingDB |
| KAT8 | p-Aminophenol | NA | 500000 | NA | NA | NA | NA | PubChem |
| KAT8 | (4-Fluorophenyl)hydrazine | NA | 310000 | NA | NA | NA | NA | BindingDB |
| KAT8 | Phenylhydrazine | NA | 1000000 | NA | NA | NA | NA | PubChem |
| KAT8 | 1,7-Cleve's acid | NA | 940000 | NA | NA | NA | NA | BindingDB |
| KAT8 | 1-Naphthylamine | NA | 181000 | NA | NA | NA | NA | BindingDB |
| KAT8 | Benzoic acid, 2-decyl-6-hydroxy- | NA | 123026877081 | NA | NA | NA | NA | BindingDB |
| KCNA1 | Bergapten | NA | NA | 200000 | NA | NA | NA | PubChem |
| KCNA1 | Flecainide | NA | 209000 | NA | NA | NA | NA | PubChem|TTD |
| KCNA1 | Diltiazem | NA | 144000 | NA | NA | NA | NA | PubChem|TTD |