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drugs and pathways
negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
KARS1
Lercanidipine
NA
320000
NA
NA
NA
NA
BindingDB
KAT2B
3-(5-Methyl-2-nitrophenoxy)propan-1-amine hydrochloride
NA
203600
NA
NA
NA
NA
TTD
KAT2B
3-(4-Chloro-2-nitrophenoxy)propan-1-amine;hydrochloride
NA
215100
NA
NA
NA
NA
TTD
KAT2B
3-(4-Methyl-2-nitrophenoxy)propan-1-amine;hydrochloride
NA
180000
NA
NA
NA
NA
TTD
KAT2B
3-(2-nitrophenoxy)propan-1-amine Hydrochloride
NA
125600
NA
NA
NA
NA
TTD
KAT2B
3-(4-Methoxy-2-nitrophenoxy)propan-1-amine;hydrochloride
NA
102700
NA
NA
NA
NA
TTD
KAT2B
4-Amino-3-methoxynaphthalen-1-ol
NA
200000
NA
NA
NA
NA
BindingDB|TTD
KAT2B
N-(4-hydroxynaphthalen-1-yl)decanamide
NA
160000
NA
NA
NA
NA
BindingDB|TTD
KAT2B
N-(4-hydroxynaphthalen-1-yl)-2-phenylacetamide
NA
500000
NA
NA
NA
NA
TTD
KAT2B
2,5-diphenylisothiazol-3(2H)-one
NA
200000
NA
NA
NA
NA
TTD
KAT2B
4-Methoxynaphthalen-1-amine hydrochloride
NA
500000
NA
NA
NA
NA
TTD
KAT2B
N-Methyl-2-(Tetrahydro-2h-Pyran-4-Yloxy)benzamide
NA
NA
104000|166000|459000
NA
NA
NA
BindingDB|ChEMBL
KAT2B
5-methyl-2-phenyl-2H-1,2,3-triazole-4-carboxamide
NA
NA
250000|360000|660000|1080000
NA
NA
NA
BindingDB|ChEMBL
KAT2B
Cambridge id 5139258
NA
145900
NA
NA
NA
NA
TTD
KAT2B
4-Nitro-1-naphthol
NA
221000
NA
NA
NA
NA
BindingDB|TTD
KAT2B
p-Aminophenol
NA
500000
NA
NA
NA
NA
PubChem|TTD
KAT2B
5-Phenylureidomethyl-2-phenylisothiazol-3(2H)-one
NA
200000
NA
NA
NA
NA
TTD
KAT2B
5-Methyl-2-N-Phenylisothiazol-3(2H)-one
NA
200000
NA
NA
NA
NA
TTD
KAT2B
4-Methoxymethyl-2-phenyl-isothiazol-3(2H)-one
NA
102000
NA
NA
NA
NA
BindingDB|TTD
KAT2B
4-Methyl-5-methoxy-2-phenyl-isothiazol-3(2H)-one
NA
200000
NA
NA
NA
NA
TTD
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