| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| JAK2 |
Tozasertib |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
1-[(1-{2-[(3-Chloro-1,2-Dimethyl-1h-Indol-5-Yl)amino]pyrimidin-4-Yl}-3-Methyl-1h-Pyrazol-4-Yl)methyl]azetidin-3-Ol |
NA |
111900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| JAK2 |
1-[(3-Methyl-1-{2-[(1,2,3-Trimethyl-1h-Indol-5-Yl)amino]pyrimidin-4-Yl}-1h-Pyrazol-4-Yl)methyl]azetidin-3-Ol |
NA |
138200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| JAK2 |
(3R)-1-[[1-[2-[(3-chloro-1,2-dimethylindol-5-yl)amino]pyrimidin-4-yl]-3-methylpyrazol-4-yl]methyl]pyrrolidin-3-ol |
NA |
162400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| JAK2 |
|
7000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
Pazopanib |
6900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- |
580000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
1-(Naphthalen-2-yl)prop-2-en-1-ol |
NA |
501000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
Benzamide, N-[6-[(6,7-dimethoxy-4-quinolinyl)oxy]-1-methyl-1H-indazol-3-yl]-3-(trifluoromethyl)- |
NA |
25000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| JAK3 |
Ast-487 |
260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
(E)-N-(4-((3-chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl)-4-(piperidin-1-yl)but-2-enamide |
NA |
3570000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| JAK3 |
1-(2-Aminoethyl)-2-piperidin-4-ylbenzimidazole-5-carboxamide |
NA |
232500 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
Ruboxistaurin |
420000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
Canertinib |
630000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
Erlotinib |
930000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
1-(6,7-Dimethoxynaphthalen-2-yl)-3-morpholin-4-ylpropan-1-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
2-Oxo-2-(3-(quinoxalin-2-yl)phenylamino)ethyl acetate |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
Sunitinib |
1200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
Jnj-7706621 |
180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| JAK3 |
Tozasertib |
630000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |