| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| JAK2 |
US10040781, Example 187 |
NA |
183000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 300 |
NA |
453000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 319 |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 355 |
NA |
474000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 369 |
NA |
718000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 455 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 454 |
NA |
621000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 456 |
NA |
966000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 457 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 518 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
1-(2-Aminoethyl)-2-piperidin-4-ylbenzimidazole-5-carboxamide |
NA |
437300 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US11279703, Table 1.1 |
NA |
359700 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
3-[4-oxo-3-(3,4,5-trifluoroanilino)-3,3a,5,6,7,7a-hexahydro-2H-pyrazolo[4,3-c]pyridin-1-yl]butanenitrile |
NA |
168700 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
3-[3-[(2-fluoropyridin-4-yl)amino]-4-oxo-3,3a,5,6,7,7a-hexahydro-2H-pyrazolo[4,3-c]pyridin-1-yl]butanenitrile |
NA |
106100 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 137 |
NA |
207000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
2-[[8-(2-Hydroxyacetyl)-8-azabicyclo[3.2.1]octan-3-yl]oxy]-5-[4-[4-[4-(oxetan-3-yl)piperazin-1-yl]anilino]-1,3-diaza-5-azoniacyclohexa-1,4,5-trien-2-yl]benzonitrile |
NA |
265000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 435 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 436 |
NA |
156000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
US10040781, Example 437 |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB |
| JAK2 |
N-[[1-[4-amino-6-(4-cyanoanilino)-1,3,5-triazin-2-yl]triazol-4-yl]methyl]methanesulfonamide |
NA |
NA |
106000 |
NA |
NA |
NA |
BindingDB |