Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| JAK2 | US10040781, Example 609 | NA | 237000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 602 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 130 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 129 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | 2-(((3R,4S)-3-fluoro-1-((4S,5S)-5-methyl-2-oxooxazolidine-4-carbonyl)piperidin-4-yl)oxy)-5-(4-((4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)amino)-1,3,5-triazin-2-yl)benzonitrile | NA | 959000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 598 | NA | 521000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 595 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 608 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 335 | NA | 478000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 606 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 601 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 596 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 594 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 607 | NA | 161000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 610 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 603 | NA | 1000000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 592 | NA | 239000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 599 | NA | 510000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 88 | NA | 488000 | NA | NA | NA | NA | BindingDB |
| JAK2 | US10040781, Example 123 | NA | 546000 | NA | NA | NA | NA | BindingDB |